3-Aminopyrrolidinone farnesyltransferase inhibitors: design of macrocyclic compounds with improved pharmacokinetics and excellent cell potency (Q24298433)

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3-Aminopyrrolidinone farnesyltransferase inhibitors: design of macrocyclic compounds with improved pharmacokinetics and excellent cell potency
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    3-Aminopyrrolidinone farnesyltransferase inhibitors: design of macrocyclic compounds with improved pharmacokinetics and excellent cell potency (English)
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    Ian M Bell
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    Steven N Gallicchio
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    Marc Abrams
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    Lorena S Beese
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    Douglas C Beshore
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    Hema Bhimnathwala
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    Michael J Bogusky
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    Carolyn A Buser
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    J Christopher Culberson
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    Joseph Davide
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    Michelle Ellis-Hutchings
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    Christine Fernandes
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    Jackson B Gibbs
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    Samuel L Graham
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    Kelly A Hamilton
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    George D Hartman
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    David C Heimbrook
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    Carl F Homnick
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    Hans E Huber
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    Joel R Huff
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    Kelem Kassahun
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    Kenneth S Koblan
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    Nancy E Kohl
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    Robert B Lobell
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    Joseph J Lynch
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    Ronald Robinson
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    A David Rodrigues
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    Jeffrey S Taylor
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    Eileen S Walsh
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    Theresa M Williams
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    C Blair Zartman
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    6 June 2002
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    45
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    12
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    2388-409
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