The pharmacology of fluparoxan: a selective α2-adrenoceptor antagonist (Q24673328)

https://api.crossref.org/works/10.1111/J.1476-5381.1991.TB12272.X

26 October 2022

1 reference

C. A. Halliday

1

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26 October 2022

B. J. Jones

2

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26 October 2022

M. Skingle

3

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26 October 2022

D. M. Walsh

4

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26 October 2022

H. Wise

5

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26 October 2022

M. B. Tyers

6

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full work available at URL

26 October 2022

language of work or name

English

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publication date

April 1991

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https://europepmc.org/articles/PMC1917968

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1677298

https://europepmc.org/articles/PMC1917968?pdf=render

26 October 2022

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A1677298

https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1111%2Fj.1476-5381.1991.tb12272.x

26 October 2022

1 reference

https://api.crossref.org/works/10.1111/J.1476-5381.1991.TB12272.X

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.1991.tb12272.x/fullpdf

26 October 2022

1 reference

https://api.crossref.org/works/10.1111/J.1476-5381.1991.TB12272.X

British Journal of Pharmacology

26 October 2022

published in

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volume

102

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issue

4

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page(s)

887-95

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

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Effects of dopamine receptor agonists and antagonists at peripheral neuronal and vascular dopamine receptors in the anaesthetised cat

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Subtypes of alpha 2-adrenoceptors: pharmacological and molecular biological evidence converge

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Receptors for 5-hydroxytryptamine and noradrenaline in rabbit isolated ear artery and aorta

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Clonidine antinociceptive activity: Effects of drugs influencing central monoaminergic and cholinergic mechanisms in the rat

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Alpha 2-adrenoceptors mediate clonidine-induced sedation in the rat.

28 September 2017

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The effects of alpha-adrenoceptor agonists and antagonists on responses of transmurally stimulated prostatic and epididymal portions of the isolated vas deferens of the rat

28 September 2017

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Pharmacological characterization of the presynaptic alpha-adrenoceptors regulating cholinergic activity in the guinea-pig ileum

28 September 2017

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The actions of some alpha-adrenoreceptor agonists and antagonists in an antinociceptive test in mice

28 September 2017

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Clonidine-induced hypoactivity and mydriasis in mice are respectively mediated via pre- and postsynaptic alpha 2-adrenoceptors in the brain

28 September 2017

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Effects of idazoxan on catecholamine systems in rat brain

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A comparison of 5-hydroxytryptamine receptors mediating contraction in rabbit aorta and dog saphenous vein: evidence for different receptor types obtained by use of selective agonists and antagonists

30 May 2018

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Pharmacological profile of a new potent and specific alpha 2-adrenoceptor antagonist, L-657,743.

30 May 2018

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(8a alpha,12a alpha,13a alpha)-5,8,8a,9,10,11,12,12a,13,13a-decahydro- 3-methoxy-12-(methylsulfonyl)-6H-isoquino[2,1-g][1,6]naphthyridi ne, a potent and highly selective alpha 2-adrenoceptor antagonist

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THE ATTRACTIONS OF PROTEINS FOR SMALL MOLECULES AND IONS

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12 December 2020

Novel and versatile superfusion system. Its use in the evaluation of some spasmogenic and spasmolytic agents using guinea-pig isolated tracheal smooth muscle

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12 December 2020

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12 December 2020

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Identifiers

0 references

PMC publication ID

1917968

0 references