Functional selectivity of dopamine D1 receptor agonists in regulating the fate of internalized receptors (Q24681428)

1

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Adam Griffith

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Scott Oloff

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Justin T Brown

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William A Goddard

6

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Richard B Mailman

Functional Selectivity and Classical Concepts of Quantitative Pharmacology

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language of work or name

English

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publication date

February 2007

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published in

Neuropharmacology

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volume

52

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issue

2

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page(s)

562-75

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cites work

1 reference

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Differential activation of adenylate cyclase and receptor internalization by novel dopamine D1 receptor agonists

7 April 2017

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Identification of a novel endocytic recycling signal in the D1 dopamine receptor

28 September 2017

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First principles predictions of the structure and function of g-protein-coupled receptors: validation for bovine rhodopsin.

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8,9-dihydroxy-1,2,3,11b-tetrahydrochromeno[4,3,2,-de]isoquinoline (dinoxyline), a high affinity and potent agonist at all dopamine receptor isoforms.

28 September 2017

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The role of phosphorylation in D1 dopamine receptor desensitization: evidence for a novel mechanism of arrestin association

28 September 2017

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The nature of the arrestin x receptor complex determines the ultimate fate of the internalized receptor

28 September 2017

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Prediction of structure and function of G protein-coupled receptors

28 September 2017

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The role of phosphorylation/dephosphorylation in agonist-induced desensitization of D1 dopamine receptor function: evidence for a novel pathway for receptor dephosphorylation.

28 September 2017

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Dinapsoline: characterization of a D1 dopamine receptor agonist in a rat model of Parkinson's disease.

28 September 2017

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Differential affinities of visual arrestin, beta arrestin1, and beta arrestin2 for G protein-coupled receptors delineate two major classes of receptors

28 September 2017

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Cellular trafficking of G protein-coupled receptor/beta-arrestin endocytic complexes

28 September 2017

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Distinct dynamin-dependent and -independent mechanisms target structurally homologous dopamine receptors to different endocytic membranes

28 September 2017

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Homologous desensitization of the D1A dopamine receptor: efficacy in causing desensitization dissociates from both receptor occupancy and functional potency.

28 September 2017

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Persistent activation of the dopamine D1 receptor contributes to prolonged receptor desensitization: studies with A-77636.

28 September 2017

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9-Dihydroxy-2,3,7,11b-tetrahydro-1H-naph[1,2,3-de]isoquinoline: a potent full dopamine D1 agonist containing a rigid-beta-phenyldopamine pharmacophore

28 September 2017

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A study of some variables in a tetrazolium dye (MTT) based assay for cell growth and chemosensitivity

28 September 2017

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A68930: a potent agonist selective for the dopamine D1 receptor

28 September 2017

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A-77636: a potent and selective dopamine D1 receptor agonist with antiparkinsonian activity in marmosets

28 September 2017

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Multiple receptors for dopamine

28 September 2017

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Femtomole sensitive radioimmunoassay for cyclic AMP and cyclic GMP after 2'0 acetylation by acetic anhydride in aqueous solution

28 September 2017

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Differential regulation of dopamine D1A receptor responsiveness by various G protein-coupled receptor kinases

28 September 2017

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Regulation of dopamine D(1) receptor trafficking by protein kinase A-dependent phosphorylation.

28 September 2017

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G(olf) and Gs in rat basal ganglia: possible involvement of G(olf) in the coupling of dopamine D1 receptor with adenylyl cyclase

30 May 2018

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Synthesis and dopaminergic activity of 3-substituted 1-(aminomethyl)-3,4-dihydro-5,6-dihydroxy-1H-2-benzopyrans: characterization of an auxiliary binding region in the D1 receptor

30 May 2018

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Comparison of the D1-dopamine agonists SKF-38393 and A-68930 in neonatal 6-hydroxydopamine-lesioned rats: behavioral effects and induction of c-fos-like immunoreactivity

30 May 2018

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Dopamine receptors: pharmacological and anatomical evidences indicate that two distinct dopamine receptor populations are present in rat striatum.

30 May 2018

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Functional selectivity, ligand-directed trafficking, conformation-specific agonism: what's in a name?

30 May 2018

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Effects of repeated dopamine D1 receptor stimulation on rotation and c-fos expression.

28 November 2018

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Conformational analysis of D1 dopamine receptor agonists: pharmacophore assessment and receptor mapping

28 November 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/17067639