Insights in 17beta-HSD1 enzyme kinetics and ligand binding by dynamic motion investigation (Q27322084)

April 2022 Public Data File from Crossref

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31 May 2018

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21 January 2018

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21 January 2018

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New insights into the SAR and binding modes of bis(hydroxyphenyl)thiophenes and -benzenes: influence of additional substituents on 17beta-hydroxysteroid dehydrogenase type 1 (17beta-HSD1) inhibitory activity and selectivity

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Elucidation of a complete kinetic mechanism for a mammalian hydroxysteroid dehydrogenase (HSD) and identification of all enzyme forms on the reaction coordinate: the example of rat liver 3alpha-HSD (AKR1C9)

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PubMed

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