Structural insights into the mode of action of a pure antiestrogen (Q27630646)

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5 November 2019

title

Structural insights into the mode of action of a pure antiestrogen (English)

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5 November 2019

1

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5 November 2019

author name string

A M Brzozowski

2

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5 November 2019

J Walton

3

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5 November 2019

R E Hubbard

4

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5 November 2019

A G Thorsell

5

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5 November 2019

Y L Li

6

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5 November 2019

J A Gustafsson

7

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5 November 2019

M Carlquist

8

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5 November 2019

publication date

1 February 2001

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5 November 2019

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5 November 2019

volume

9

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5 November 2019

issue

2

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5 November 2019

page(s)

145-153

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The steroid and thyroid hormone receptor superfamily

5 November 2019

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Response to a specific antioestrogen (ICI 182780) in tamoxifen-resistant breast cancer

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Estrogen receptor (ER) modulators each induce distinct conformational changes in ER alpha and ER beta.

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Inhibition of estrogen receptor-DNA binding by the "pure" antiestrogen ICI 164,384 appears to be mediated by impaired receptor dimerization

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7 January 2021

The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen

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7 January 2021

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist

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Identifiers

DOI

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5 November 2019

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