2-Amino-3,4-dihydroquinazolines as inhibitors of BACE-1 (beta-site APP cleaving enzyme): Use of structure based design to convert a micromolar hit into a nanomolar lead (Q27647023)

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2-Amino-3,4-dihydroquinazolines as inhibitors of BACE-1 (beta-site APP cleaving enzyme): Use of structure based design to convert a micromolar hit into a nanomolar lead
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    2-Amino-3,4-dihydroquinazolines as inhibitors of BACE-1 (beta-site APP cleaving enzyme): Use of structure based design to convert a micromolar hit into a nanomolar lead (English)
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    Ellen W Baxter
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    Kelly A Conway
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    Ludo Kennis
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    François Bischoff
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    Marc H Mercken
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    Charles H Reynolds
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    Brett A Tounge
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    Chi Luo
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    Malcolm K Scott
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    Yifang Huang
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    Mirielle Braeken
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    Serge M A Pieters
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    Didier J C Berthelot
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    Stefan Masure
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    Wouter D Bruinzeel
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    Alfonzo D Jordan
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    Robert E Boyd
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    Junya Qu
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    Richard S Alexander
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    Douglas E Brenneman
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    Allen B Reitz
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    6 September 2007
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    50
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    18
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    4261-4
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