Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo model (Q27650834)

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Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo model
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    Discovery of novel, potent benzamide inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1) exhibiting oral activity in an enzyme inhibition ex vivo model (English)
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    Lisa D Julian
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    Zhulun Wang
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    Tracy Bostick
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    Seb Caille
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    Rebekah Choi
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    Michael DeGraffenreid
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    Yongmei Di
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    Xiao He
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    Randall W Hungate
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    Juan C Jaen
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    Jinsong Liu
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    Mario Monshouwer
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    Dustin McMinn
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    Yosup Rew
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    Athena Sudom
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    Hua Tu
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    Stefania Ursu
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    Nigel Walker
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    Jay P Powers
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    10 July 2008
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    51
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    13
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    3953-60
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