Discovery of (R)-6-cyclopentyl-6-(2-(2,6-diethylpyridin-4-yl)ethyl)-3-((5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl)-4-hydroxy-5,6-dihydropyran-2-one (PF-00868554) as a potent and orally available hepatitis C virus polymerase inhibitor (Q27653726)

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Discovery of (R)-6-cyclopentyl-6-(2-(2,6-diethylpyridin-4-yl)ethyl)-3-((5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl)-4-hydroxy-5,6-dihydropyran-2-one (PF-00868554) as a potent and orally available hepatitis C virus polymerase inhibitor
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    Discovery of (R)-6-cyclopentyl-6-(2-(2,6-diethylpyridin-4-yl)ethyl)-3-((5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)methyl)-4-hydroxy-5,6-dihydropyran-2-one (PF-00868554) as a potent and orally available hepatitis C virus polymerase inhibitor (English)
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    Hui Li
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    John Tatlock
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    Angelica Linton
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    Javier Gonzalez
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    Tanya Jewell
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    Leena Patel
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    Sarah Ludlum
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    Matthew Drowns
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    Sadayappan V Rahavendran
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    Heather Skor
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    Robert Hunter
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    Stephanie T Shi
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    Koleen J Herlihy
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    Hans Parge
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    Michael Hickey
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    Xiu Yu
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    Fannie Chau
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    Cristina Lewis
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    12 March 2009
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    52
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    5
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    1255-8
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