Peptide Length and Leaving-Group Sterics Influence Potency of Peptide Phosphonate Protease Inhibitors (Q27666756)

2

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Aura A Eroy-Reveles

3

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Pascal Egea

4

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Cheryl Tajon

5

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Charles S Craik

MEROPS: the peptidase database

6

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publication date

28 January 2011

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published in

Chemistry and Biology

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volume

18

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issue

1

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page(s)

48-57

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cites work

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Combination treatment with VELCADE and low-dose tissue plasminogen activator provides potent neuroprotection in aged rats after embolic focal ischemia

20 March 2017

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27 November 2018

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27 November 2018

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Synthesis and evaluation of diphenyl phosphonate esters as inhibitors of the trypsin-like granzymes A and K and mast cell tryptase

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Dipeptide phosphonates as inhibitors of dipeptidyl peptidase IV

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Amino acid and peptide phosphonate derivatives as specific inhibitors of serine peptidases

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Novel amidine-containing peptidyl phosphonates as irreversible inhibitors for blood coagulation and related serine proteases

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Inhibition of trypsin and urokinase by Cbz-amino(4-guanidinophenyl)methanephosphonate aromatic ester derivatives: the influence of the ester group on their biological activity

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Irreversible inhibition of serine proteases by peptide derivatives of (alpha-aminoalkyl)phosphonate diphenyl esters

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12 December 2020