A selective, orally bioavailable 1,2,4-triazolo[1,5-a]pyridine-based inhibitor of Janus kinase 2 for use in anticancer therapy: discovery of CEP-33779 (Q27679143)

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A selective, orally bioavailable 1,2,4-triazolo[1,5-a]pyridine-based inhibitor of Janus kinase 2 for use in anticancer therapy: discovery of CEP-33779
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    A selective, orally bioavailable 1,2,4-triazolo[1,5-a]pyridine-based inhibitor of Janus kinase 2 for use in anticancer therapy: discovery of CEP-33779 (English)
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    Benjamin J Dugan
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    Diane E Gingrich
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    Eugen F Mesaros
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    Karen L Milkiewicz
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    Matthew A Curry
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    Allison L Zulli
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    Pawel Dobrzanski
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    Cynthia Serdikoff
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    Mahfuza Jan
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    Thelma S Angeles
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    Mark S Albom
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    Jennifer L Mason
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    Lisa D Aimone
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    Sheryl L Meyer
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    Zeqi Huang
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    Kevin J Wells-Knecht
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    Mark A Ator
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    Bruce A Ruggeri
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    Bruce D Dorsey
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    14 June 2012
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    55
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    11
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    5243-54
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