Discovery of 7-methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (GSK2606414), a potent and selective first-in-class inhibitor of protein kinase R (PKR)-like endoplasmic reticulum kinase (P (Q27681837)
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| Language | Label | Description | Also known as |
|---|---|---|---|
| English | Discovery of 7-methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (GSK2606414), a potent and selective first-in-class inhibitor of protein kinase R (PKR)-like endoplasmic reticulum kinase (P |
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Statements
Discovery of 7-methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (GSK2606414), a potent and selective first-in-class inhibitor of protein kinase R (PKR)-like endoplasmic reticulum kinase (PERK) (English)
Jeffrey M Axten
Jesús R Medina
Yanhong Feng
Arthur Shu
Stuart P Romeril
Seth W Grant
William Hoi Hong Li
Dirk A Heerding
Elisabeth Minthorn
Thomas Mencken
Charity Atkins
Qi Liu
Sridhar Rabindran
Rakesh Kumar
Xuan Hong
Aaron Goetz
Thomas Stanley
Scott D Sigethy
Ginger H Tomberlin
Annie M Hassell
Kirsten M Kahler
Lisa M Shewchuk
8 August 2012
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