X-ray Structural and Biological Evaluation of a Series of Potent and Highly Selective Inhibitors of Human Coronavirus Papain-like Proteases (Q27681891)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24568342%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

7

Susan C Baker

1 reference

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7 June 2020

5

Anna M Mielech

1 reference

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7 June 2020

1

Yahira M Báez-Santos

1 reference

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7 June 2020

8

Scott D Larsen

1 reference

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7 June 2020

author name string

Scott J Barraza

2

1 reference

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7 June 2020

Michael W Wilson

3

1 reference

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7 June 2020

Michael P Agius

4

1 reference

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7 June 2020

Nicole M Davis

6

1 reference

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Journal of Medicinal Chemistry

7 June 2020

language of work or name

English

0 references

publication date

27 March 2014

0 references

published in

1 reference

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7 June 2020

volume

57

1 reference

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7 June 2020

issue

6

1 reference

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7 June 2020

page(s)

2393-2412

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24568342%20AND%20SRC:MED&resulttype=core&format=json

Middle East respiratory syndrome coronavirus (MERS-CoV): announcement of the Coronavirus Study Group

7 June 2020

cites work

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20 March 2017

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20 March 2017

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The papain-like protease from the severe acute respiratory syndrome coronavirus is a deubiquitinating enzyme

20 March 2017

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An efficient one-step site-directed and site-saturation mutagenesis protocol

20 March 2017

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Synergistic inhibitor binding to the papain-like protease of human SARS coronavirus: mechanistic and inhibitor design implications

7 April 2017

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Novel inhibitors of bacterial virulence: development of 5,6-dihydrobenzo[h]quinazolin-4(3H)-ones for the inhibition of group A streptococcal streptokinase expression

29 September 2017

1 reference

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Human coronavirus EMC is not the same as severe acute respiratory syndrome coronavirus

29 September 2017

1 reference

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Genomic characterization of a newly discovered coronavirus associated with acute respiratory distress syndrome in humans

29 September 2017

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Severe respiratory illness caused by a novel coronavirus, in a patient transferred to the United Kingdom from the Middle East, September 2012.

29 September 2017

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Coronavirus papain-like proteases negatively regulate antiviral innate immune response through disruption of STING-mediated signaling

29 September 2017

1 reference

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Structure-based design, synthesis, and biological evaluation of a series of novel and reversible inhibitors for the severe acute respiratory syndrome-coronavirus papain-like protease

29 September 2017

1 reference

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Drug targets in severe acute respiratory syndrome (SARS) virus and other coronavirus infections

29 September 2017

1 reference

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A noncovalent class of papain-like protease/deubiquitinase inhibitors blocks SARS virus replication

29 September 2017

1 reference

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Regulation of IRF-3-dependent innate immunity by the papain-like protease domain of the severe acute respiratory syndrome coronavirus

29 September 2017

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Severe acute respiratory syndrome coronavirus papain-like protease: structure of a viral deubiquitinating enzyme

29 September 2017

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The papain-like protease of severe acute respiratory syndrome coronavirus has deubiquitinating activity

29 September 2017

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Identification of severe acute respiratory syndrome coronavirus replicase products and characterization of papain-like protease activity

29 September 2017

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The synthesis and biology of fluorinated prostacyclins

29 September 2017

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Interaction of methylenedioxyphenyl (1,3-benzodioxole) compounds with enzymes and their effects on mammals.

29 September 2017

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2 June 2018

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27 November 2018

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27 November 2018

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27 November 2018

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Selectivity in ISG15 and ubiquitin recognition by the SARS coronavirus papain-like protease

27 November 2018

1 reference

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The binding of HIV-1 protease inhibitors to human serum proteins

27 November 2018

1 reference

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Determination of serum protein binding affinity of inhibitors from analysis of concentration-response plots in biochemical activity assays

27 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24568342

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Mechanism of the metabolism of 1,3-benzodioxoles to carbon monoxide

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24568342

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM401712T

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24568342%20AND%20SRC:MED&resulttype=core&format=json

release_cjsqfmclq5guxfdy6exb4xnkbi

7 June 2020

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/cjsqfmclq5guxfdy6exb4xnkbi

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24568342%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24568342%20AND%20SRC:MED&resulttype=core&format=json