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    Discovery and preclinical profile of teneligliptin (3-[(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]pyrrolidin-2-ylcarbonyl]thiazolidine): a highly potent, selective, long-lasting and orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes (English)
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    Tomohiro Yoshida
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    Fumihiko Akahoshi
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    Hiroshi Sakashita
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    Hiroshi Kitajima
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    Mitsuharu Nakamura
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    Shuji Sonda
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    Masahiro Takeuchi
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    Yoshihito Tanaka
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    Naoko Ueda
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    Sumie Sekiguchi
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    Takayuki Ishige
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    Kyoko Shima
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    Mika Nabeno
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    Yuji Abe
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    Jun Anabuki
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    Aki Soejima
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    Kumiko Yoshida
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    Yoko Takashina
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    Shinichi Ishii
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    Satoko Kiuchi
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    Sayaka Fukuda
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    Reiko Tsutsumiuchi
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    Keigo Kosaka
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    Takahiro Murozono
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    Yoshinobu Nakamaru
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    Hiroyuki Utsumi
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    Naoya Masutomi
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    Hiroyuki Kishida
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    Ikuko Miyaguchi
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    Yoshiharu Hayashi
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    1 October 2012
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    20
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    19
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    5705-19
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