Tebipenem, a New Carbapenem Antibiotic, Is a Slow Substrate That Inhibits the β-Lactamase from Mycobacterium tuberculosis (Q27683862)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

title

Tebipenem, a new carbapenem antibiotic, is a slow substrate that inhibits the β-lactamase from Mycobacterium tuberculosis (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

Mycobacterium tuberculosis

18 March 2020

main subject

carbapenem antibiotic

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1

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18 March 2020

3

John S Blanchard

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

author name string

Hua Xu

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

language of work or name

English

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publication date

29 May 2014

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

volume

53

1 reference

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18 March 2020

page(s)

3671-3678

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18 March 2020

issue

22

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

NXL104 Irreversibly Inhibits the β-Lactamase from Mycobacterium tuberculosis

18 March 2020

cites work

1 reference

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Structures of the Michaelis Complex (1.2 Å) and the Covalent Acyl Intermediate (2.0 Å) of Cefamandole Bound in the Active Sites of the Mycobacterium tuberculosis β-Lactamase K73A and E166A Mutants,

20 March 2017

1 reference

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Biochemical and Structural Characterization of Mycobacterium tuberculosis β-Lactamase with the Carbapenems Ertapenem and Doripenem

20 March 2017

1 reference

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20 March 2017

1 reference

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Meropenem-Clavulanate Is Effective Against Extensively Drug-Resistant Mycobacterium tuberculosis

20 March 2017

1 reference

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Multimodular penicillin-binding proteins: an enigmatic family of orthologs and paralogs

20 March 2017

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Effect of beta-lactamase location in Escherichia coli on penicillin synergy

20 March 2017

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20 March 2017

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Refinement of macromolecular structures by the maximum-likelihood method

20 March 2017

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A graphical user interface to the CCP4 program suite

20 March 2017

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Incorporation of prior phase information strengthens maximum-likelihood structure refinement

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4053071

Intestinal absorption mechanism of tebipenem pivoxil, a novel oral carbapenem: involvement of human OATP family in apical membrane transport

7 April 2017

1 reference

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The chemical biology of new drugs in the development for tuberculosis

29 September 2017

1 reference

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Current status of newer carbapenems

29 September 2017

1 reference

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Bacterial resistance to beta-lactam antibiotics: compelling opportunism, compelling opportunity

29 September 2017

1 reference

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Appropriate prescribing of oral beta-lactam antibiotics.

29 September 2017

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In vitro antibacterial activity of LJC 11,036, an active metabolite of L-084, a new oral carbapenem antibiotic with potent antipneumococcal activity

29 September 2017

1 reference

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Progress in global tuberculosis control 1995-1996, with emphasis on 22 high-incidence countries. Global Monitoring and Surveillance Project.

29 September 2017

1 reference

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Irreversible inhibition of the Mycobacterium tuberculosis beta-lactamase by clavulanate

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4053071

Clinical use of the meropenem-clavulanate combination for extensively drug-resistant tuberculosis.

2 June 2018

1 reference

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Pharmacokinetics of tebipenem pivoxil, a novel oral carbapenem antibiotic, in experimental animals

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4053071

Population pharmacokinetics of tebipenem pivoxil (ME1211), a novel oral carbapenem antibiotic, in pediatric patients with otolaryngological infection or pneumonia

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4053071

Genetic analysis of the beta-lactamases of Mycobacterium tuberculosis and Mycobacterium smegmatis and susceptibility to beta-lactam antibiotics

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4053071

Revised Ambler classification of {beta}-lactamases

27 November 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24846409

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Processing of X-ray diffraction data collected in oscillation mode

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24846409

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/BI500339J

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json

18 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24846409%20AND%20SRC:MED&resulttype=core&format=json