Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973) (Q27684146)

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Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973)
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    Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973) (English)
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    Kenneth D Rice
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    Naing Aay
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    Neel K Anand
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    Charles M Blazey
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    Owen J Bowles
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    Joerg Bussenius
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    Simona Costanzo
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    Jeffry K Curtis
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    Steven C Defina
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    Larisa Dubenko
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    Stefan Engst
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    Anagha A Joshi
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    Abigail R Kennedy
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    Angie I Kim
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    Elena S Koltun
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    Julie C Lougheed
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    Jean-Claire L Manalo
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    Jean-Francois Martini
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    John M Nuss
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    Csaba J Peto
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    Tsze H Tsang
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    Peiwen Yu
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    Stuart Johnston
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    10 May 2012
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    3
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    5
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    416-21
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