New substrate analogues of human serotonin N-acetyltransferase produce in situ specific and potent inhibitors (Q28238260)

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17 November 2019

title

New substrate analogues of human serotonin N-acetyltransferase produce in situ specific and potent inhibitors (English)

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17 November 2019

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14

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17 November 2019

Jean A Boutin

16

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17 November 2019

author name string

Gilles Ferry

1

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17 November 2019

Caroline Ubeaud

2

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17 November 2019

Julien Mozo

3

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17 November 2019

Christophe Péan

4

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17 November 2019

Philippe Hennig

5

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17 November 2019

Marianne Rodriguez

6

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17 November 2019

Catherine Scoul

7

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17 November 2019

Anne Bonnaud

8

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17 November 2019

Olivier Nosjean

9

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17 November 2019

Jean-Pierre Galizzi

10

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17 November 2019

Philippe Delagrange

11

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17 November 2019

Pierre Renard

12

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17 November 2019

Jean-Paul Volland

13

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17 November 2019

Daniel Lesieur

15

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17 November 2019

language of work or name

English

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publication date

1 January 2004

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17 November 2019

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17 November 2019

volume

271

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17 November 2019

issue

2

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17 November 2019

page(s)

418-428

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The human serotonin N-acetyltransferase (EC 2.3.1.87) gene (AANAT): structure, chromosomal localization, and tissue expression

17 November 2019

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Substrate specificity and inhibition studies of human serotonin N-acetyltransferase

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Structure-activity relationships for substrates and inhibitors of pineal 5-hydroxytryptamine-N-acetyltransferase: preliminary studies

21 April 2017

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Mechanism-based inhibition of the melatonin rhythm enzyme: pharmacologic exploitation of active site functional plasticity

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X-ray crystallographic studies of serotonin N-acetyltransferase catalysis and inhibition

21 April 2017

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A Potent Inhibitor of the Melatonin Rhythm Enzyme

21 April 2017

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Role of a pineal cAMP-operated arylalkylamine N-acetyltransferase/14-3-3-binding switch in melatonin synthesis

21 April 2017

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Kinetic analysis of the catalytic mechanism of serotonin N-acetyltransferase (EC 2.3.1.87)

21 April 2017

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A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

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Involvement of the mt1 melatonin receptor in human breast cancer

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Effect of melatonin on bone metabolism in ovariectomized rats

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Characterization and regulation of a CHO cell line stably expressing human serotonin N-acetyltransferase (EC 2.3.1.87).

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Bisubstrate ketone analogues as serotonin N-acetyltransferase inhibitors

21 January 2018

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Synthesis of 2-amido-2,3-dihydro-1H-phenalene derivatives as new conformationally restricted ligands for melatonin receptors

21 January 2018

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Synthesis of phenalene and acenaphthene derivatives as new conformationally restricted ligands for melatonin receptors

21 January 2018

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Melatonergic properties of the (+)- and (-)-enantiomers of N-(4-methoxy-2,3-dihydro-1H-phenalen-2-yl)amide derivatives

21 January 2018

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Synthesis of a small library of phenylalkylamide derivatives as melatoninergic ligands for human mt1 and MT2 receptors.

21 January 2018

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Synthesis and structure-affinity-activity relationships of novel benzofuran derivatives as MT(2) melatonin receptor selective ligands

21 January 2018

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Control of melatonin synthesis in the mammalian pineal gland: the critical role of serotonin acetylation

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Serotonin N-acetyltransferase: mechanism and inhibition

21 January 2018

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Synthesis and structure-activity relationships of novel naphthalenic and bioisosteric related amidic derivatives as melatonin receptor ligands

21 January 2018

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Tetrahydronaphthalenic derivatives as new agonist and antagonist ligands for melatonin receptors

21 January 2018

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Substituted oxygenated heterocycles and thio-analogues: synthesis and biological evaluation as melatonin ligands

21 January 2018

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