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    Discovery of a Plasmodium falciparum glucose-6-phosphate dehydrogenase 6-phosphogluconolactonase inhibitor (R,Z)-N-((1-ethylpyrrolidin-2-yl)methyl)-2-(2-fluorobenzylidene)-3-oxo-3,4-dihydro-2H-benzo[b][1,4]thiazine-6-carboxamide (ML276) that reduces parasite growth in vitro (English)
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    Janina Preuss
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    Patrick Maloney
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    Satyamaheshwar Peddibhotla
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    Michael P Hedrick
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    Paul Hershberger
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    Palak Gosalia
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    Monika Milewski
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    Yujie Linda Li
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    Eliot Sugarman
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    Becky Hood
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    Eigo Suyama
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    Kevin Nguyen
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    Stefan Vasile
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    Eduard Sergienko
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    Arianna Mangravita-Novo
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    Michael Vicchiarelli
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    Danielle McAnally
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    Gregory P Roth
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    Jena Diwan
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    Thomas D Y Chung
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    Esther Jortzik
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    Stefan Rahlfs
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    Lars Bode
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    23 August 2012
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    55
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    16
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    7262-72
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