Sulfotransferase structural biology and inhibitor discovery (Q28295987)

Crystal structure of estrogen sulphotransferase

Europe PubMed Central

title

Sulfotransferase structural biology and inhibitor discovery (English)

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Virginia L Rath

1

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Dawn Verdugo

series ordinal

2

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Stefan Hemmerich

series ordinal

3

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language of work or name

English

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publication date

1 December 2004

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published in

Drug Discovery Today

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volume

9

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issue

23

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page(s)

1003-11

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cites work

1 reference

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7 January 2021

Structure of a human carcinogen-converting enzyme, SULT1A1. Structural and kinetic implications of substrate inhibition

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7 January 2021

Crystal structure of human catecholamine sulfotransferase

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Crystal structure of human cholesterol sulfotransferase (SULT2B1b) in the presence of pregnenolone and 3'-phosphoadenosine 5'-phosphate. Rationale for specificity differences between prototypical SULT2A1 and the SULT2BG1 isoforms

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7 January 2021

Identification, function and structure of the mycobacterial sulfotransferase that initiates sulfolipid-1 biosynthesis

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7 January 2021

Crystal structure of the sulfotransferase domain of human heparan sulfate N-deacetylase/ N-sulfotransferase 1

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Crystal structure and mutational analysis of heparan sulfate 3-O-sulfotransferase isoform 1.

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Strategies for drug discovery by targeting sulfation pathways

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Conserved structural motifs in the sulfotransferase family

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Glivec (STI571, imatinib), a rationally developed, targeted anticancer drug

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The sulfuryl transfer mechanism. Crystal structure of a vanadate complex of estrogen sulfotransferase and mutational analysis

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7 January 2021

Identification of amino acid residues critical for catalysis and cosubstrate binding in the flavonol 3-sulfotransferase

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7 January 2021

Structural basis of lectin-carbohydrate recognition

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Biosynthesis of L-selectin ligands: sulfation of sialyl Lewis x-related oligosaccharides by a family of GlcNAc-6-sulfotransferases

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Sulfation of N-acetylglucosamine by chondroitin 6-sulfotransferase 2 (GST-5).

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Identification of an N-acetylglucosamine-6-0-sulfotransferase activity specific to lymphoid tissue: an enzyme with a possible role in lymphocyte homing

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Potent inhibition of estrogen sulfotransferase by hydroxylated PCB metabolites: a novel pathway explaining the estrogenic activity of PCBs

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IV. Synthesis and assay of analogs of adenosine 3',5'-diphosphate as inhibitors of bovine adrenal estrogen sulfotranferase

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A library approach to the generation of bisubstrate analogue sulfotransferase inhibitors

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Synthesis of a bisubstrate analogue targeting estrogen sulfotransferase

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Discovery of estrogen sulfotransferase inhibitors from a purine library screen

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In vitro sulfotransferase activity of NodH, a nodulation protein of Rhizobium meliloti required for host-specific nodulation

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Discovery of Carbohydrate Sulfotransferase Inhibitors from a Kinase-Directed Library We thank Sharon Long and Dave Keating for providing both the NodH sulfotransferase and APS Kinase during our preliminary experiments and Jack Kirsch for [...]

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Synthesis and application of functionally diverse 2,6,9-trisubstituted purine libraries as CDK inhibitors

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Crystal structures of catalytic subunit of cAMP-dependent protein kinase in complex with isoquinolinesulfonyl protein kinase inhibitors H7, H8, and H89. Structural implications for selectivity

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Tyrosylprotein sulfotransferase inhibitors generated by combinatorial target-guided ligand assembly

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10.1016/S1359-6446(04)03273-8

Identifiers

DOI

1 reference

Consolidated OpenCitations Corpus – April 2017

1 reference

Consolidated OpenCitations Corpus – April 2017

PubMed publication ID

15574316

1 reference

Consolidated OpenCitations Corpus – April 2017