Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor (Q28300800)

PubMed ID

8987785

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8987785%20AND%20SRC:MED&resulttype=core&format=json

22 October 2019

title

Bicuculline and gabazine are allosteric inhibitors of channel opening of the GABAA receptor (English)

1 reference

PubMed ID

8987785

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8987785%20AND%20SRC:MED&resulttype=core&format=json

22 October 2019

1 reference

3

C Zorumski

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=PMCID:PMC6573228&resulttype=core&format=json

15 May 2020

author name string

S Ueno

1

1 reference

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15 May 2020

J Bracamontes

2

1 reference

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15 May 2020

D S Weiss

4

1 reference

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15 May 2020

J H Steinbach

5

1 reference

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15 May 2020

language of work or name

English

0 references

publication date

1 January 1997

1 reference

PubMed ID

8987785

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8987785%20AND%20SRC:MED&resulttype=core&format=json

22 October 2019

published in

Journal of Neuroscience

1 reference

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15 May 2020

volume

17

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15 May 2020

issue

2

1 reference

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15 May 2020

page(s)

625-634

1 reference

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Mutagenesis of the 43-kD postsynaptic protein defines domains involved in plasma membrane targeting and AChR clustering

15 May 2020

cites work

1 reference

12 December 2020

Neurosteroid analogues: structure-activity studies of benz[e]indene modulators of GABAA receptor function. 1. The effect of 6-methyl substitution on the electrophysiological activity of 7-substituted benz[e]indene-3-carbonitriles

1 reference

12 December 2020

Multiple mechanisms of antagonism of gamma-aminobutyric acid (GABA) responses

1 reference

12 December 2020

Potentiation of gamma-aminobutyric-acid-activated chloride conductance by a steroid anaesthetic in cultured rat spinal neurones

1 reference

12 December 2020

The effects of pentobarbital and related compounds on frog motoneurons

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12 December 2020

Visual identification of individual transfected cells for electrophysiology using antibody-coated beads

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Propofol activates GABAA receptor-chloride ionophore complex in dissociated hippocampal pyramidal neurons of the rat.

1 reference

12 December 2020

Quantitative evaluation of the properties of a pyridazinyl GABA derivative (SR 95531) as a GABAA competitive antagonist. An electrophysiological approach.

1 reference

12 December 2020

Kinetic properties of the pentobarbitone-gated chloride current in frog sensory neurones

1 reference

12 December 2020

Endogenous subunits can cause ambiguities in the pharmacology of exogenous gamma-aminobutyric acidA receptors expressed in human embryonic kidney 293 cells

1 reference

12 December 2020

GABAA receptor needs two homologous domains of the beta-subunit for activation by GABA but not by pentobarbital.

1 reference

12 December 2020

Point mutations affecting antagonist affinity and agonist dependent gating of GABAA receptor channels.

1 reference

12 December 2020

Intraburst kinetic properties of the GABAA receptor main conductance state of mouse spinal cord neurones in culture

1 reference

12 December 2020

A novel GABAA antagonist [3H]SR 95531: microscopic analysis of binding in the rat brain and allosteric modulation by several benzodiazepine and barbiturate receptor ligands.

1 reference

12 December 2020

High-efficiency transformation of mammalian cells by plasmid DNA

1 reference

12 December 2020

Modulation of the GABAA receptor by depressant barbiturates and pregnane steroids

1 reference

12 December 2020

Differences in the expression of GABA(A) receptors between functionally innervated and non-innervated granule neurons in neonatal rat cerebellar cultures.

1 reference

12 December 2020

GABA antagonists differentiate between recombinant GABAA/benzodiazepine receptor subtypes

1 reference

12 December 2020

Desensitized states prolong GABAA channel responses to brief agonist pulses.

1 reference

12 December 2020

GABA-dependent modulation of the Cl- ionophore by steroids in rat brain.

1 reference

12 December 2020

Barbiturate interactions at the human GABAA receptor: dependence on receptor subunit combination

1 reference

12 December 2020

GABAA receptor channels

1 reference

12 December 2020

Chloride current induced by alcohols in rat dorsal root ganglion neurons

1 reference

12 December 2020

Volatile anesthetics gate a chloride current in postnatal rat hippocampal neurons

1 reference

12 December 2020

Improved patch-clamp techniques for high-resolution current recording from cells and cell-free membrane patches

1 reference

12 December 2020

Barbiturates allosterically inhibit GABA antagonist and benzodiazepine inverse agonist binding

1 reference

12 December 2020

Drug blockade of open end-plate channels

1 reference

12 December 2020

How quickly can GABAA receptors open?

1 reference

12 December 2020

Mutations affecting the glycine receptor agonist transduction mechanism convert the competitive antagonist, picrotoxin, into an allosteric potentiator.

1 reference

12 December 2020

Effects of a benz[e]indene on gamma-aminobutyric acid-gated chloride currents in cultured postnatal rat hippocampal neurons

1 reference

12 December 2020

10.1523/JNEUROSCI.17-02-00625.1997

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=PMCID:PMC6573228&resulttype=core&format=json

OpenCitations bibliographic resource ID

15 May 2020

3373901

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=PMCID:PMC6573228&resulttype=core&format=json

15 May 2020

2 references

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

3373901