Interaction of batrachotoxin with the local anesthetic receptor site in transmembrane segment IVS6 of the voltage-gated sodium channel (Q28369249)

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A R Cantrell

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Y Qu

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T Scheuer

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W A Catterall

Proceedings of the National Academy of Sciences of the United States of America

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language of work or name

English

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publication date

10 November 1998

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published in

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volume

95

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issue

23

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page(s)

13947-52

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cites work

Point mutations in segment I-S6 render voltage-gated Na+ channels resistant to batrachotoxin

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Common molecular determinants of local anesthetic, antiarrhythmic, and anticonvulsant block of voltage-gated Na+ channels

20 March 2017

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Improved patch-clamp techniques for high-resolution current recording from cells and cell-free membrane patches

20 March 2017

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Molecular determinants of drug binding and action on L-type calcium channels

20 March 2017

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A unique role for the S4 segment of domain 4 in the inactivation of sodium channels

29 September 2017

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Structure and function of voltage-dependent sodium channels: comparison of brain II and cardiac isoforms

29 September 2017

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Molecular determinants of high affinity binding of alpha-scorpion toxin and sea anemone toxin in the S3-S4 extracellular loop in domain IV of the Na+ channel alpha subunit

29 September 2017

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Transfecting mammalian cells: optimization of critical parameters affecting calcium-phosphate precipitate formation

29 September 2017

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Fast lidocaine block of cardiac and skeletal muscle sodium channels: one site with two routes of access.

29 September 2017

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Modification of cardiac Na+ channels by batrachotoxin: effects on gating, kinetics, and local anesthetic binding

29 September 2017

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

A mutation in segment IVS6 disrupts fast inactivation of sodium channels

29 September 2017

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Structure and function of voltage-gated ion channels

29 September 2017

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Neurotoxins that Act on Voltage-Sensitive Sodium Channels in Excitable Membranes

29 September 2017

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Batrachotoxin: chemistry and pharmacology

29 September 2017

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A molecular view of neurotransmitter receptors and ionic channels

29 September 2017

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An integrated view of the molecular toxinology of sodium channel gating in excitable cells

29 September 2017

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Batrachotoxin as a tool to study voltage-sensitive sodium channels of excitable membranes

29 September 2017

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Molecular mechanisms of local anesthesia: a review

29 September 2017

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Receptor sites for Ca2+ channel antagonists

29 September 2017

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Sea anemone toxin and scorpion toxin share a common receptor site associated with the action potential sodium ionophore

29 September 2017

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Class I antiarrhythmic drugs: allosteric inhibitors of [3H] batrachotoxinin binding to rat cardiac sodium channels.

29 September 2017

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Molecular determinants of state-dependent block of Na+ channels by local anesthetics

2 June 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Modification of cloned brain Na+ channels by batrachotoxin

2 June 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Functional co-expression of the beta 1 and type IIA alpha subunits of sodium channels in a mammalian cell line

2 June 2018

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Panning transfected cells for electrophysiological studies

2 June 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Batrachotoxin-induced depolarization and [3H]batrachotoxinin-a 20 alpha-benzoate binding in a vesicular preparation from guinea pig cerebral cortex

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Binding of batrachotoxinin A 20-alpha-benzoate to a receptor site associated with sodium channels in synaptic nerve ending particles

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Activation of the action potential Na+ ionophore by neurotoxins. An allosteric model

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Dopaminergic modulation of sodium current in hippocampal neurons via cAMP-dependent phosphorylation of specific sites in the sodium channel alpha subunit.

2 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Neurotoxin binding and allosteric modulation at receptor sites 2 and 5 on purified and reconstituted rat brain sodium channels.

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Modulation of cardiac Na+ channel expression in Xenopus oocytes by beta 1 subunits.

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Inhibition of binding of [3H]batrachotoxinin A 20-alpha-benzoate to sodium channels by local anesthetics

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Pyrethroid insecticides: stereospecific allosteric interaction with the batrachotoxinin-A benzoate binding site of mammalian voltage-sensitive sodium channels.

27 November 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=24981

Cellular and molecular biology of voltage-gated sodium channels

27 November 2018

1 reference

12 December 2020

Interaction of insecticides of the pyrethroid family with specific binding sites on the voltage-dependent sodium channel from mammalian brain

1 reference

12 December 2020

Further analysis of the mechanisms of action of batrachotoxin on the membrane of myelinated nerve

1 reference

12 December 2020

Toxin T4(6) from Ptychodiscus brevis (formerly Gymnodinium breve) enhances activation of voltage-sensitive sodium channels by veratridine

1 reference

12 December 2020

Inhibition of voltage-sensitive sodium channels in neuroblastoma cells by antiarrhythmic drugs

1 reference

12 December 2020

Inhibition of binding of [3H]batrachotoxinin A 20-alpha-benzoate to sodium channels by the anticonvulsant drugs diphenylhydantoin and carbamazepine

1 reference

12 December 2020

Visual identification of individual transfected cells for electrophysiology using antibody-coated beads

1 reference

12 December 2020

Site of covalent labeling by a photoreactive batrachotoxin derivative near transmembrane segment IS6 of the sodium channel alpha subunit

1 reference

12 December 2020

Depth asymmetries of the pore-lining segments of the Na+ channel revealed by cysteine mutagenesis

1 reference

12 December 2020