Discovery of diverse small molecule chemotypes with cell-based PKD1 inhibitory activity (Q28477356)

21 June 2017

title

Discovery of diverse small molecule chemotypes with cell-based PKD1 inhibitory activity (English)

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21 June 2017

1 reference

Robyn B Reed

6

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John S. Lazo

series ordinal

10

object named as

John S Lazo

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21 June 2017

9

Peter Wipf

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21 June 2017

1

Elizabeth R Sharlow

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21 June 2017

4

Stephanie Leimgruber

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21 June 2017

7

Tong Ying Shun

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21 June 2017

Gabriela Mustata Wilson

series ordinal

2

object named as

Gabriela Mustata Wilson

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21 June 2017

3

David Close

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5

Manuj Tandon

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21 June 2017

Q Jane Wang

8

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21 June 2017

language of work or name

English

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publication date

5 October 2011

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21 June 2017

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21 June 2017

volume

6

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issue

10

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21 June 2017

page(s)

e25134

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Creative Commons Attribution 4.0 International

21 June 2017

copyright license

start time

5 October 2011

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April 2022 Public Data File from Crossref

copyright status

copyrighted

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cites work

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Characterization of the biological effects of a novel protein kinase D inhibitor in endothelial cells

19 March 2017

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Comparative surface geometry of the protein kinase family

19 March 2017

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Identification of protein kinase D2 as a pivotal regulator of endothelial cell proliferation, migration, and angiogenesis

19 March 2017

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Protein kinase D-dependent phosphorylation and nuclear export of histone deacetylase 5 mediates vascular endothelial growth factor-induced gene expression and angiogenesis

19 March 2017

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Role of the regulatory domain of protein kinase D2 in phorbol ester binding, catalytic activity, and nucleocytoplasmic shuttling

19 March 2017

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Manipulation of alternative splicing by a newly developed inhibitor of Clks

19 March 2017

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Synthesis and Structure-Activity Relationships of Benzothienothiazepinone Inhibitors of Protein Kinase D

19 March 2017

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Protein kinase D signaling: multiple biological functions in health and disease

29 September 2017

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A novel protein kinase D inhibitor attenuates early events of experimental pancreatitis in isolated rat acini

29 September 2017

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Protein kinase D2 is a crucial regulator of tumour cell-endothelial cell communication in gastrointestinal tumours

29 September 2017

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Novel protein kinase D inhibitors cause potent arrest in prostate cancer cell growth and motility

29 September 2017

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A novel small-molecule inhibitor of protein kinase D blocks pancreatic cancer growth in vitro and in vivo

29 September 2017

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Profiling the NIH Small Molecule Repository for compounds that generate H2O2 by redox cycling in reducing environments

29 September 2017

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Potent and selective disruption of protein kinase D functionality by a benzoxoloazepinolone

29 September 2017

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Development, validation and implementation of immobilized metal affinity for phosphochemicals (IMAP)-based high-throughput screening assays for low-molecular-weight compound libraries

29 September 2017

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Protein kinase D3 (PKD3) contributes to prostate cancer cell growth and survival through a PKCepsilon/PKD3 pathway downstream of Akt and ERK 1/2.

29 September 2017

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Protein kinase d in the cardiovascular system: emerging roles in health and disease.

29 September 2017

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Development and implementation of a miniaturized high-throughput time-resolved fluorescence energy transfer assay to identify small molecule inhibitors of polo-like kinase 1.

29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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Expression of the protein kinase D (PKD) family during mouse embryogenesis

29 September 2017

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Isoquinolinesulfonamides, novel and potent inhibitors of cyclic nucleotide-dependent protein kinase and protein kinase C

2 June 2018

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Vascular endothelial growth factor induces protein kinase D-dependent production of proinflammatory cytokines in endothelial cells.

2 June 2018

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Protein kinase C nu/protein kinase D3 nuclear localization, catalytic activation, and intracellular redistribution in response to G protein-coupled receptor agonists

21 January 2018

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The activation loop phosphorylation of protein kinase D is an early marker of neuronal DNA damage.

21 January 2018

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Epigenetic inactivation of protein kinase D1 in gastric cancer and its role in gastric cancer cell migration and invasion

21 January 2018

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Identification of Orally Available Naphthyridine Protein Kinase D Inhibitors

21 January 2018

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Identification of Potent and Selective Amidobipyridyl Inhibitors of Protein Kinase D

21 January 2018

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A novel kinase inhibitor establishes a predominant role for protein kinase D as a cardiac class IIa histone deacetylase kinase

21 January 2018

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3,5-diarylazoles as novel and selective inhibitors of protein kinase D.

21 January 2018

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10.1371/JOURNAL.PONE.0025134

21 January 2018

Identifiers

DOI

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21 June 2017

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