Identification of compounds with anti-proliferative activity against Trypanosoma brucei brucei strain 427 by a whole cell viability based HTS campaign (Q28485372)

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English	Identification of compounds with anti-proliferative activity against Trypanosoma brucei brucei strain 427 by a whole cell viability based HTS campaign	scientific article

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19 February 2020

Identification of compounds with anti-proliferative activity against Trypanosoma brucei brucei strain 427 by a whole cell viability based HTS campaign (English)

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19 February 2020

infectious disease

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Trypanosoma brucei

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1

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19 February 2020

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19 February 2020

Jean-Robert Ioset

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Jean-Robert Ioset

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19 February 2020

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Jonathan B Baell

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19 February 2020

Eric Chatelain

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19 February 2020

Sarah R Moawad

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19 February 2020

Danny Ganame

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29 November 2012

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19 February 2020

PLoS Neglected Tropical Diseases

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19 February 2020

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19 February 2020

11

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19 February 2020

e1896

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19 February 2020

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Creative Commons Attribution 4.0 International

29 November 2012

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SCYX-7158, an orally-active benzoxaborole for the treatment of stage 2 human African trypanosomiasis

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The mitochondrion is a site of trypanocidal action of the aromatic diamidine DB75 in bloodstream forms of Trypanosoma brucei

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A chromosomal SIR2 homologue with both histone NAD-dependent ADP-ribosyltransferase and deacetylase activities is involved in DNA repair in Trypanosoma brucei

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12 December 2020

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12 December 2020

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1 reference

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12 December 2020

based on heuristic

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1 reference

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10.1371/JOURNAL.PNTD.0001896

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Consolidated OpenCitations Corpus – April 2017

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