Structural and energetic effects of A2A adenosine receptor mutations on agonist and antagonist binding (Q28543560)

April 2022 Public Data File from Crossref

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The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

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Molecular mechanisms of ligand binding, signaling, and regulation within the superfamily of G-protein-coupled receptors: molecular modeling and mutagenesis approaches to receptor structure and function

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Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognition

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Hydration Site Thermodynamics Explain SARs for Triazolylpurines Analogues Binding to the A2A Receptor

7 April 2017

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