Molecular basis for selectivity of high affinity peptide antagonists for the gastrin-releasing peptide receptor (Q28568038)

1

1 reference

31 January 2017

T. Katsuno

2

1 reference

31 January 2017

S. J. Hocart

3

1 reference

31 January 2017

D. H. Coy

4

1 reference

31 January 2017

M. Llinares

5

1 reference

31 January 2017

R. T. Jensen

Journal of Biological Chemistry

7

1 reference

31 January 2017

language of work or name

English

0 references

publication date

28 September 2001

1 reference

31 January 2017

1 reference

31 January 2017

276

1 reference

31 January 2017

39

1 reference

31 January 2017

36652–36663

1 reference

31 January 2017

Mammalian bombesin receptors

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Progress in the development of potent bombesin receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Bombesin receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Effects of potent bombesin antagonist on exocrine pancreatic secretion in rats

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Role of bombesin-related peptides in the control of food intake

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Role of vagal fibers and bombesin/gastrin-releasing peptide-neurons in distention-induced gastrin release in rats.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Inhibition of growth of OV-1063 human epithelial ovarian cancers and c- jun and c- fos oncogene expression by bombesin antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Tyrosine 220 in the 5th transmembrane domain of the neuromedin B receptor is critical for the high selectivity of the peptoid antagonist PD168368.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Delineation of a region in the B2 bradykinin receptor that is essential for high-affinity agonist binding

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Bombesin-induction of cell proliferation in 3T3 cells. Specific receptors and early signaling events

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Neuroendocrine dysdifferentiation and bombesin production in carcinogen-induced hepatocellular rat tumours

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Interaction of bombesin and related peptides with receptors on pancreatic acinar cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Bombesin: potential integrative peptide for feeding and satiety

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Bombesin: central nervous system actions to affect the autonomic nervous system

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Molecular cloning of the bombesin/gastrin-releasing peptide receptor from Swiss 3T3 cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

cDNA cloning, characterization, and brain region-specific expression of a neuromedin-B-preferring bombesin receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Two distinct receptor subtypes for mammalian bombesin-like peptides

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Syntheses and biological activities of potent bombesin receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

JMV641: a potent bombesin receptor antagonist that inhibits Swiss 3T3 cell proliferation

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Lipofection: a highly efficient, lipid-mediated DNA-transfection procedure

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Ligand binding, internalization, degradation and regulation by guanine nucleotides of bombesin receptor subtypes: a comparative study

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

LIGAND: A versatile computerized approach for characterization of ligand-binding systems

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

GPCRDB: an information system for G protein-coupled receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

21 January 2018

The Protein Data Bank

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Structural analysis based on state-space modeling

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Protein classification by stochastic modeling and optimal filtering of amino-acid sequences.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

SWISS-MODEL and the Swiss-PdbViewer: an environment for comparative protein modeling

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Calculation of conformational ensembles from potentials of mean force. An approach to the knowledge-based prediction of local structures in globular proteins.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Cloning and expression of the neuromedin B receptor and the third subtype of bombesin receptor genes in the mouse

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

The 'peptoid' approach to the design of non-peptide, small molecule agonists and antagonists of neuropeptides

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

A single amino acid of the cholecystokinin-B/gastrin receptor determines specificity for non-peptide antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Arginine 336 and asparagine 333 of the human cholecystokinin-A receptor binding site interact with the penultimate aspartic acid and the C-terminal amide of cholecystokinin.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Separable binding sites for the natural agonist endothelin-1 and the non-peptide antagonist bosentan on human endothelin-A receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Development of potent gastrin-releasing peptide antagonists having a D-Pro-psi(CH2NH)-Phe-NH2 C terminus

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Role of the extracellular domains of the cholecystokinin receptor in agonist binding.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Mutation of aspartate residues in the third extracellular loop of the rat B2 bradykinin receptor decreases affinity for bradykinin

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Modeling the G-protein-coupled neuropeptide Y Y1 receptor agonist and antagonist binding sites.

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Amino acids of the third transmembrane domain of the AT1A angiotensin II receptor are involved in the differential recognition of peptide and nonpeptide ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Cation-pi interactions in chemistry and biology: a new view of benzene, Phe, Tyr, and Trp

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200

Crystal structure of rhodopsin: A G protein-coupled receptor

21 January 2018

1 reference

https://api.crossref.org/works/10.1074%2FJBC.M104566200