Molecular mechanism of action of monocyclam versus bicyclam non-peptide antagonists in the CXCR4 chemokine receptor (Q30832371)

27 June 2017

title

Molecular mechanism of action of monocyclam versus bicyclam non-peptide antagonists in the CXCR4 chemokine receptor (English)

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27 June 2017

Mette M Rosenkilde

1

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Thue W Schwartz

object named as

Thue W Schwartz

7

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Dominique Schols

object named as

Dominique Schols

5

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author name string

Lars-Ole Gerlach

2

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27 June 2017

Sigrid Hatse

3

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27 June 2017

Renato T Skerlj

4

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Gary J Bridger

6

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27 June 2017

language of work or name

English

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publication date

28 June 2007

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Journal of Biological Chemistry

27 June 2017

published in

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27 June 2017

volume

282

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27 June 2017

issue

37

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27 June 2017

page(s)

27354-27365

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Expression pattern of HIV-1 coreceptors on T cells: implications for viral transmission and lymphocyte homing

27 June 2017

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21 January 2018

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Synthesis and structure-activity relationships of phenylenebis(methylene)-linked bis-azamacrocycles that inhibit HIV-1 and HIV-2 replication by antagonism of the chemokine receptor CXCR4

21 January 2018

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Metal ion enhanced binding of AMD3100 to Asp262 in the CXCR4 receptor

21 January 2018

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Synthesis and structure-activity relationships of phenylenebis(methylene)-linked bis-tetraazamacrocycles that inhibit HIV replication. Effects of macrocyclic ring size and substituents on the aromatic linker

21 January 2018

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Synthesis and structure-activity relationships of phenylenebis(methylene)-linked bis-tetraazamacrocycles that inhibit human immunodeficiency virus replication. 2. Effect of heteroaromatic linkers on the activity of bicyclams

21 January 2018

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Highly potent and selective inhibition of human immunodeficiency virus by the bicyclam derivative JM3100

21 January 2018

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Quantitative structural activity relationship study of bis-tetraazacyclic compounds. A novel series of HIV-1 and HIV-2 inhibitors

21 January 2018

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AMD3100 mobilizes hematopoietic stem cells with long-term repopulating capacity in nonhuman primates.

21 January 2018

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21 January 2018

Identifiers

DOI

10.1074/JBC.M704739200

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27 June 2017

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