Discovery of (R)-7-cyano-2,3,4, 5-tetrahydro-1-(1H-imidazol-4-ylmethyl)-3- (phenylmethyl)-4-(2-thienylsulfonyl)-1H-1,4-benzodiazepine (BMS-214662), a farnesyltransferase inhibitor with potent preclinical antitumor activity (Q31445193)
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English | Discovery of (R)-7-cyano-2,3,4, 5-tetrahydro-1-(1H-imidazol-4-ylmethyl)-3- (phenylmethyl)-4-(2-thienylsulfonyl)-1H-1,4-benzodiazepine (BMS-214662), a farnesyltransferase inhibitor with potent preclinical antitumor activity |
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Discovery of (R)-7-cyano-2,3,4, 5-tetrahydro-1-(1H-imidazol-4-ylmethyl)-3- (phenylmethyl)-4-(2-thienylsulfonyl)-1H-1,4-benzodiazepine (BMS-214662), a farnesyltransferase inhibitor with potent preclinical antitumor activity (English)
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Hunt JT
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Ding CZ
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Batorsky R
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Bednarz M
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Bhide R
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Cho Y
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Chong S
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Chao S
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Gullo-Brown J
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Guo P
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Kim SH
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Lee FY
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Leftheris K
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Miller A
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Mitt T
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Patel M
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Penhallow BA
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Ricca C
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Rose WC
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Schmidt R
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Slusarchyk WA
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Vite G
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Manne V
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