First-line treatment for chronic myeloid leukemia: dasatinib, nilotinib, or imatinib (Q33392977)

26 July 2017

5 references

3 April 2019

2 August 2019

17 September 2019

5 December 2020

17 December 2020

First-line treatment for chronic myeloid leukemia: dasatinib, nilotinib, or imatinib (English)

1 reference

26 July 2017

main subject

chronic myeloid leukemia

3 references

3 April 2019

2 August 2019

17 September 2019

1 reference

2 August 2019

heterocyclic compound

1 reference

17 September 2019

1 reference

1 reference

5 December 2020

1 reference

17 December 2020

dasatinib monohydrate

1 reference

1 reference

1 reference

Guoqing Wei

1

1 reference

26 July 2017

Shamudheen Rafiyath

series ordinal

2

1 reference

26 July 2017

Delong Liu

series ordinal

3

1 reference

26 July 2017

language of work or name

English

1 reference

National Center for Biotechnology Information

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/esummary.fcgi?db=pubmed&retmode=json&id=21108851

3 September 2024

publication date

26 November 2010

6 references

full work available at URL

26 July 2017

3 April 2019

2 August 2019

17 September 2019

5 December 2020

17 December 2020

https://jhoonline.biomedcentral.com/counter/pdf/10.1186/1756-8722-3-47

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

http://www.jhoonline.org/content/3//47

3 September 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

http://www.jhoonline.org/content/3//47/abstract

3 September 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

http://www.jhoonline.org/content/pdf/1756-8722-3-47.pdf

3 September 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

https://www.ncbi.nlm.nih.gov/pmc/articles/pmid/21108851/?tool=EBI

3 September 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

https://www.ncbi.nlm.nih.gov/pmc/articles/pmid/21108851/pdf/?tool=EBI

3 September 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

https://europepmc.org/articles/PMC3000369

3 September 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

https://europepmc.org/articles/PMC3000369?pdf=render

3 September 2024

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A21108851

https://link.springer.com/content/pdf/10.1186/1756-8722-3-47.pdf

3 September 2024

1 reference

https://api.crossref.org/works/10.1186/1756-8722-3-47

Journal of Hematology & Oncology

3 September 2024

published in

6 references

26 July 2017

3 April 2019

2 August 2019

17 September 2019

5 December 2020

17 December 2020

3

1 reference

26 July 2017

page(s)

47

1 reference

Creative Commons Attribution 2.0 Generic

26 July 2017

copyright license

5 references

3 April 2019

2 August 2019

17 September 2019

5 December 2020

on focus list of Wikimedia project

17 December 2020

copyright status

copyrighted

0 references

ScienceSource

0 references

cites work

Nilotinib versus imatinib for newly diagnosed chronic myeloid leukemia

1 reference

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First-line therapy for chronic myeloid leukemia: new horizons and an update

21 June 2018

1 reference

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Tyrosine kinase inhibitors: the first decade

21 June 2018

1 reference

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Novel therapeutic agents against cancer stem cells of chronic myeloid leukemia

21 June 2018

1 reference

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Danusertib (formerly PHA-739358)--a novel combined pan-Aurora kinases and third generation Bcr-Abl tyrosine kinase inhibitor

21 June 2018

1 reference

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Phase III, randomized, open-label study of daily imatinib mesylate 400 mg versus 800 mg in patients with newly diagnosed, previously untreated chronic myeloid leukemia in chronic phase using molecular end points: tyrosine kinase inhibitor optimizati

21 June 2018

1 reference

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Nilotinib as front-line treatment for patients with chronic myeloid leukemia in early chronic phase

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Results of dasatinib therapy in patients with early chronic-phase chronic myeloid leukemia

21 June 2018

1 reference

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Severe toxicity of skin rash, fever and diarrhea associated with imatinib: case report and review of skin toxicities associated with tyrosine kinase inhibitors.

21 June 2018

1 reference

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The occurrence and management of fluid retention associated with TKI therapy in CML, with a focus on dasatinib

21 June 2018

1 reference

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AP24534, a pan-BCR-ABL inhibitor for chronic myeloid leukemia, potently inhibits the T315I mutant and overcomes mutation-based resistance

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

The new tyrosine-kinase inhibitor and anticancer drug dasatinib reversibly affects platelet activation in vitro and in vivo.

21 June 2018

1 reference

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Inhibitory effects of omacetaxine on leukemic stem cells and BCR-ABL-induced chronic myeloid leukemia and acute lymphoblastic leukemia in mice

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Bleeding diathesis in patients with chronic myelogenous leukemia receiving dasatinib therapy

21 June 2018

1 reference

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New dosing schedules of dasatinib for CML and adverse event management

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Characteristics and outcomes of patients with chronic myeloid leukemia and T315I mutation following failure of imatinib mesylate therapy

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Simultaneous targeting of Aurora kinases and Bcr-Abl kinase by the small molecule inhibitor PHA-739358 is effective against imatinib-resistant BCR-ABL mutations including T315I.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Congestive heart failure is a rare event in patients receiving imatinib therapy

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

In vitro and in vivo activity of SKI-606, a novel Src-Abl inhibitor, against imatinib-resistant Bcr-Abl+ neoplastic cells

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Cardiotoxicity of the cancer therapeutic agent imatinib mesylate.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Nilotinib in imatinib-resistant CML and Philadelphia chromosome-positive ALL

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Comparison of imatinib mesylate, dasatinib (BMS-354825), and nilotinib (AMN107) in an N-ethyl-N-nitrosourea (ENU)-based mutagenesis screen: high efficacy of drug combinations

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

The structure of Dasatinib (BMS-354825) bound to activated ABL kinase domain elucidates its inhibitory activity against imatinib-resistant ABL mutants

21 June 2018

1 reference

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21 June 2018

Adherence to Medication

1 reference

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In vitro activity of Bcr-Abl inhibitors AMN107 and BMS-354825 against clinically relevant imatinib-resistant Abl kinase domain mutants

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Characterization of AMN107, a selective inhibitor of native and mutant Bcr-Abl.

21 June 2018

1 reference

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Imatinib compared with interferon and low-dose cytarabine for newly diagnosed chronic-phase chronic myeloid leukemia

21 June 2018

1 reference

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Genetic variation in bilirubin UPD-glucuronosyltransferase gene promoter and Gilbert's syndrome

21 June 2018

1 reference

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The genetic basis of the reduced expression of bilirubin UDP-glucuronosyltransferase 1 in Gilbert's syndrome

21 June 2018

1 reference

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Dasatinib versus imatinib in newly diagnosed chronic-phase chronic myeloid leukemia

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Adherence is the critical factor for achieving molecular responses in patients with chronic myeloid leukemia who achieve complete cytogenetic responses on imatinib.

31 October 2018

1 reference

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New developments in tyrosine kinase inhibitor therapy for newly diagnosed chronic myeloid leukemia

31 October 2018

1 reference

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Nilotinib for the frontline treatment of Ph(+) chronic myeloid leukemia

31 October 2018

1 reference

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Prevalence, determinants, and outcomes of nonadherence to imatinib therapy in patients with chronic myeloid leukemia: the ADAGIO study.

31 October 2018

1 reference

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Activity of bosutinib, dasatinib, and nilotinib against 18 imatinib-resistant BCR/ABL mutants

31 October 2018

1 reference

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Finding of kinase domain mutations in patients with chronic phase chronic myeloid leukemia responding to imatinib may identify those at high risk of disease progression

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Omacetaxine mepesuccinate--a semisynthetic formulation of the natural antitumoral alkaloid homoharringtonine, for chronic myelocytic leukemia and other myeloid malignancies.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Solution conformations and dynamics of ABL kinase-inhibitor complexes determined by NMR substantiate the different binding modes of imatinib/nilotinib and dasatinib

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Cardiac events in imatinib mesylate-treated chronic myeloid leukemia patients: A single institution experience

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

Resistance to dasatinib in Philadelphia-positive leukemia patients and the presence or the selection of mutations at residues 315 and 317 in the BCR-ABL kinase domain

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3000369

UGT1A1 promoter polymorphism increases risk of nilotinib-induced hyperbilirubinemia

31 October 2018

1 reference

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Mutation status and clinical outcome of 89 imatinib mesylate-resistant chronic myelogenous leukemia patients: a retrospective analysis from the French intergroup of CML (Fi(phi)-LMC GROUP)

31 October 2018

1 reference

12 December 2020

Treatment interruptions and non-adherence with imatinib and associated healthcare costs: a retrospective analysis among managed care patients with chronic myelogenous leukaemia

1 reference

12 December 2020

MK-0457, a novel kinase inhibitor, is active in patients with chronic myeloid leukemia or acute lymphocytic leukemia with the T315I BCR-ABL mutation

1 reference

12 December 2020

Clinical outcome of 27 imatinib mesylate-resistant chronic myelogenous leukemia patients harboring a T315I BCR-ABL mutation

1 reference

12 December 2020

In reply to 'Cardiotoxicity of the cancer therapeutic agent imatinib mesylate'

1 reference

12 December 2020

Drug Design, Development and Therapy

24

2

215

X Huang

2008

1 reference

https://api.crossref.org/works/10.1186/1756-8722-3-47

3 September 2024

36

1

e4

Z Xu

2009

1 reference

https://api.crossref.org/works/10.1186/1756-8722-3-47

3 September 2024

54

93

47

P Shah

2008

1 reference

https://api.crossref.org/works/10.1186/1756-8722-3-47

3 September 2024

Identifiers

1 reference

Dimensions Publication ID

26 July 2017

1 reference

https://scigraph.springernature.com/pub.10.1186/1756-8722-3-47

9 September 2019

1 reference

26 July 2017

1 reference