Characterization and optimization of a red-shifted fluorescence polarization ADP detection assay (Q33404831)

26 July 2017

title

Characterization and optimization of a red-shifted fluorescence polarization ADP detection assay (English)

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26 July 2017

Karen M Kleman-Leyer

1

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26 July 2017

Tony A Klink

2

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26 July 2017

Andrew L Kopp

3

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26 July 2017

Thane A Westermeyer

4

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26 July 2017

Mark D Koeff

5

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26 July 2017

Brad R Larson

6

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26 July 2017

Tracy J Worzella

7

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26 July 2017

Cori A Pinchard

8

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26 July 2017

Sebastianus A T van de Kar

9

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26 July 2017

Guido J R Zaman

10

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26 July 2017

Jorrit J Hornberg

11

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26 July 2017

Robert G Lowery

12

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26 July 2017

publication date

1 February 2009

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Assay and Drug Development Technologies

26 July 2017

published in

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26 July 2017

volume

7

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26 July 2017

issue

1

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26 July 2017

page(s)

56-67

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Fluorescence spectroscopic profiling of compound libraries

26 July 2017

cites work

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Development of a Transcreener kinase assay for protein kinase A and demonstration of concordance of data with a filter-binding assay format

21 June 2018

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Targeted covalent inactivation of protein kinases by resorcylic acid lactone polyketides.

21 June 2018

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Transcreener: screening enzymes involved in covalent regulation

21 June 2018

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Features of selective kinase inhibitors

21 June 2018

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Discovery and characterization of a substrate selective p38alpha inhibitor

21 June 2018

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Overcoming compound interference in fluorescence polarization-based kinase assays using far-red tracers

21 June 2018

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21 June 2018

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Isozyme-nonselective N-substituted bipiperidylcarboxamide acetyl-CoA carboxylase inhibitors reduce tissue malonyl-CoA concentrations, inhibit fatty acid synthesis, and increase fatty acid oxidation in cultured cells and in experimental animals

21 June 2018

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Beta galactosidase enzyme fragment complementation as a novel technology for high throughput screening

21 June 2018

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Fluorescence assays for high-throughput screening of protein kinases

21 June 2018

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Issues and progress with protein kinase inhibitors for cancer treatment

21 June 2018

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Designing screens: how to make your hits a hit.

21 June 2018

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Protein kinases--the major drug targets of the twenty-first century?

21 June 2018

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Multiplexed enzyme assays in capillary electrophoretic single-use microfluidic devices

21 June 2018

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Determination of nucleotides and sugar nucleotides involved in protein glycosylation by high-performance anion-exchange chromatography: sugar nucleotide contents in cultured insect cells and mammalian cells

21 June 2018

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Protein kinases as therapeutic targets

21 June 2018

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A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 June 2018

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A synthetic inhibitor of the mitogen-activated protein kinase cascade

21 June 2018

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Evaluating PI3 kinase isoforms using Transcreener ADP assays

21 June 2018

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A generic, homogenous method for measuring kinase and inhibitor activity via adenosine 5'-diphosphate accumulation

31 October 2018

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A Robot-based platform to measure multiple enzyme activities in Arabidopsis using a set of cycling assays: comparison of changes of enzyme activities and transcript levels during diurnal cycles and in prolonged darkness

31 October 2018

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Identification of kinase inhibitors by an ATP depletion method

31 October 2018

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High-throughput screening with quantitation of ATP consumption: a universal non-radioisotope, homogeneous assay for protein kinase

31 October 2018

1 reference

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A homogeneous fluorescence polarization assay adaptable for a range of protein serine/threonine and tyrosine kinases

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2956686

BMS-345541 is a highly selective inhibitor of I kappa B kinase that binds at an allosteric site of the enzyme and blocks NF-kappa B-dependent transcription in mice

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2956686

Determination of 5-AMP in the presence of excess 3'(2')-AMP with the aid of antibodies raised against n6-carboxymethyl-5'-AMP conjugates. Use for the quantitation of pyridine nucleotides and of protein-bound ADP-ribose

31 October 2018

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12 December 2020

Preparation of cyclic nucleotide antisera with thyroglobulin-cyclic nucleotide conjugates

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12 December 2020

Effect of pressure on antigen-antibody complexes: modulation by temperature and ionic strength

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12 December 2020

Discovery of acetyl-coenzyme A carboxylase 2 inhibitors: comparison of a fluorescence intensity-based phosphate assay and a fluorescence polarization-based ADP Assay for high-throughput screening

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12 December 2020

Role of salt bridge formation in antigen-antibody interaction. Entropic contribution to the complex between hen egg white lysozyme and its monoclonal antibody HyHEL10

1 reference

12 December 2020

Identifiers

DOI

10.1089/ADT.2008.175

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26 July 2017

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26 July 2017

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