The Rhodadyns, a New Class of Small Molecule Inhibitors of Dynamin GTPase Activity (Q33630482)

28 July 2017

title

The Rhodadyns, a New Class of Small Molecule Inhibitors of Dynamin GTPase Activity (English)

1 reference

28 July 2017

Lisa von Kleist

8

0 references

Mark Robertson

Mark J Robertson

1

0 references

Volker Haucke

Volker Haucke

10

0 references

Adam McCluskey

Adam McCluskey

12

0 references

Phillip J. Robinson

Phillip J Robinson

11

0 references

Ngoc Chau

9

Ngoc Chau

1 reference

28 July 2017

Gordana Hadzic

2

1 reference

28 July 2017

Joseph Ambrus

3

1 reference

28 July 2017

D Yuri Pomè

4

1 reference

28 July 2017

Emily Hyde

5

1 reference

28 July 2017

Ainslie Whiting

6

1 reference

28 July 2017

Anna Mariana

7

1 reference

28 July 2017

language of work or name

1 reference

26 March 2012

1 reference

ACS Medicinal Chemistry Letters

28 July 2017

published in

1 reference

28 July 2017

volume

3

1 reference

28 July 2017

issue

5

1 reference

28 July 2017

page(s)

352-356

1 reference

Role of the clathrin terminal domain in regulating coated pit dynamics revealed by small molecule inhibition

28 July 2017

cites work

1 reference

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Molecular mechanism and physiological functions of clathrin-mediated endocytosis

21 June 2018

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The pthaladyns: GTP competitive inhibitors of dynamin I and II GTPase derived from virtual screening

21 June 2018

1 reference

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Iminochromene inhibitors of dynamins I and II GTPase activity and endocytosis

21 June 2018

1 reference

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Privileged scaffolds for library design and drug discovery

21 June 2018

1 reference

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Suppression of dynamin GTPase activity by sertraline leads to inhibition of dynamin-dependent endocytosis.

21 June 2018

1 reference

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Inhibition of dynamin mediated endocytosis by the dynoles--synthesis and functional activity of a family of indoles

21 June 2018

1 reference

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Rhodanine as a privileged scaffold in drug discovery

21 June 2018

1 reference

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Azido and diazarinyl analogues of bis-tyrphostin as asymmetrical inhibitors of dynamin GTPase

21 June 2018

1 reference

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Dynasore, a cell-permeable inhibitor of dynamin

21 June 2018

1 reference

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Bacterial entry into cells: a role for the endocytic machinery

21 June 2018

1 reference

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Small molecule inhibitors of dynamin I GTPase activity: development of dimeric tyrphostins

21 June 2018

1 reference

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Mutations in dynamin 2 cause dominant centronuclear myopathy

21 June 2018

1 reference

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Listeria hijacks the clathrin-dependent endocytic machinery to invade mammalian cells

21 June 2018

1 reference

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Mutations in the pleckstrin homology domain of dynamin 2 cause dominant intermediate Charcot-Marie-Tooth disease

21 June 2018

1 reference

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Involvement of Clathrin-Mediated Endocytosis in Human Immunodeficiency Virus Type 1 Entry

21 June 2018

1 reference

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Dynamin I phosphorylation and the control of synaptic vesicle endocytosis.

21 June 2018

1 reference

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The dynamin superfamily: universal membrane tubulation and fission molecules?

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Insider information: what viruses tell us about endocytosis

21 June 2018

1 reference

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Traffic jams II: an update of diseases of intracellular transport

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

OPA1 (Kjer type) dominant optic atrophy: a novel mitochondrial disease.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Traffic jam: a compendium of human diseases that affect intracellular transport processes

21 June 2018

1 reference

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Dynamin and its role in membrane fission

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

OPA1, encoding a dynamin-related GTPase, is mutated in autosomal dominant optic atrophy linked to chromosome 3q28

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Differential distribution of dynamin isoforms in mammalian cells

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

The dynamins: redundant or distinct functions for an expanding family of related GTPases?

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Localization of dynamin: widespread distribution in mature neurons and association with membranous organelles

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Multiple forms of dynamin are encoded by shibire, a Drosophila gene involved in endocytosis

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Dynamin-like protein encoded by the Drosophila shibire gene associated with vesicular traffic

21 June 2018

1 reference

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Depolarization-induced phosphorylation of specific proteins, mediated by calcium ion influx, in rat brain synaptosomes

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Differential phosphorylation of dynamin I isoforms in subcellular compartments demonstrates the hidden complexity of phosphoproteomes

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Some selective serotonin reuptake inhibitors inhibit dynamin I guanosine triphosphatase (GTPase).

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Myristyl Trimethyl Ammonium Bromide and Octadecyl Trimethyl Ammonium Bromide Are Surface-Active Small Molecule Dynamin Inhibitors that Block Endocytosis Mediated by Dynamin I or Dynamin II

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Dynamin GTPase regulated by protein kinase C phosphorylation in nerve terminals

30 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4025782

Protein phosphorylation is required for endocytosis in nerve terminals: potential role for the dephosphins dynamin I and synaptojanin, but not AP180 or amphiphysin

30 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24900478

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Dynamin and endocytosis

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24900478

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML200284S

1 reference

release_rg7nt3oidzatjkh3z644j6mlzi

28 July 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/rg7nt3oidzatjkh3z644j6mlzi

mapped directly with Wikidata item

24 November 2022

based on heuristic

PMC publication ID

4025782

1 reference

28 July 2017

1 reference