Enantiomers of bronchodilating beta2-adrenoceptor agonists: is there a cause for concern? (Q33636114)

28 July 2017

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title

Enantiomers of bronchodilating beta2-adrenoceptor agonists: is there a cause for concern? (English)

1 reference

28 July 2017

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Waldeck B

1

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PubMed ID

10329804

28 July 2017

language of work or name

English

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publication date

1 May 1999

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The Journal of Allergy and Clinical Immunology

28 July 2017

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28 July 2017

103

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28 July 2017

5 Pt 1

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28 July 2017

742-748

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Physiological consequences of β-adrenoceptor desensitization in guinea pigs

28 July 2017

1 reference

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7 January 2021

Chronic exposure to a β2-adrenoceptor agonist increases the airway response to methacholine

1 reference

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7 January 2021

Chronic fenoterol exposure increases in vivo and in vitro airway responses in guinea pigs

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Rebound increase in bronchial responsiveness after treatment with inhaled terbutaline

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Regular inhaled salbutamol and airway responsiveness to allergen

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Active enantiomers may cause adverse effects in asthma

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Sympathomimetic enantiomers and asthma

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Steric aspects of agonism and antagonism at beta-adrenoceptors: synthesis of and pharmacological experiments with the enantiomers of formoterol and their diastereomers

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Salbutamol in the treatment of asthma

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Biological significance of the enantiomeric purity of drugs

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Absolute configuration of the optical isomers of salbutamol

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Resolution of terbutaline, a new -sympathomimetic amine

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Some observations on the -adrenoceptor agonist properties of the isomers of salbutamol

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Steric Aspects of Agonism and Antagonism at β-Adrenoceptors: Experiments with the Enantiomers of Terbutaline and Pindolol

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

The effects of formoterol, a long-acting beta 2-adrenoceptor agonist, on mucociliary activity

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

The pharmacology of salmeterol

1 reference

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7 January 2021

Steric aspects of agonism and antagonism at beta-adrenoceptors: experiments with the enantiomers of clenbuterol

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Atypical molecular pharmacology of a new long-acting beta 2-adrenoceptor agonist, TA 2005

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Comparison of R-, S-, and RS-albuterol interaction with human beta 1- and beta 2-adrenergic receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Effects of the enantiomers of R,S-salbutamol on incompletely fused tetanic contractions of slow- and fast-twitch skeletal muscles of the guinea-pig

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Airway hyperreactivity.

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Increased airway reactivity in the guinea-pig follows exposure to intravenous isoprenaline.

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Enhancement of airway reactivity to histamine by isoprenaline and related beta-adrenoceptor agonists in the guinea-pig.

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Hyperresponsiveness of the airways following exposure of guinea-pigs to racemic mixtures and distomers of beta 2-selective sympathomimetics.

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Effects of albuterol enantiomers on in vitro bronchial reactivity

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Effects of S-salbutamol on human isolated bronchus

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Steric aspects of formoterol and terbutaline: is there an adverse effect of the distomer on airway smooth muscle function?

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

S-albuterol exacerbates calcium responses to carbachol in airway smooth muscle cells

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

(S)-Albuterol increases intracellular free calcium by muscarinic receptor activation and a phospholipase C-dependent mechanism in airway smooth muscle.

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Do parasympatholytic effects of long-acting beta 2-sympathomimetics contribute to their relaxant effects in airway smooth muscle cells?

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Effect of enantiomeric forms of albuterol on stimulated secretion of granular protein from human eosinophils

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Beta-adrenergic regulation of the eosinophil respiratory burst as detected by lucigenin-dependent luminescence

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Beta-adrenoceptor agonists block corticosteroid inhibition in eosinophils

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Differential responses of asthmatic airways to enantiomers of albuterol. Implications for clinical treatment of asthma

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Effect of single doses of S-salbutamol, R-salbutamol, racemic salbutamol, and placebo on the airway response to methacholine

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Pharmacokinetics and extrapulmonary beta 2 adrenoceptor activity of nebulised racemic salbutamol and its R and S isomers in healthy volunteers

1 reference

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7 January 2021

Improved bronchodilation with levalbuterol compared with racemic albuterol in patients with asthma

1 reference

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7 January 2021

The debate on S-enantiomers of beta-agonists: tempest in a teapot or gathering storm?

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Tracheal Relaxing Effects and β2-Selectivity of TA-2005, a Newly Developed Bronchodilating Agent, in Isolated Guinea Pig Tissues

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Picumeterol: dissociation of improvement in lung function and reduction of airways hyperresponsiveness in asthmatics

1 reference

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7 January 2021

Stereochemistry, a basis for sophisticated nonsense in pharmacokinetics and clinical pharmacology

1 reference

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7 January 2021

Analysis of salbutamol enantiomers in human urine by chiral high-performance liquid chromatography and preliminary studies related to the stereoselective disposition kinetics in man

1 reference

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7 January 2021

Enantioselective disposition of salbutamol in man following oral and intravenous administration

1 reference

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7 January 2021

Stereoselective sulphate conjugation of salbutamol in humans: comparison of hepatic, intestinal and platelet activity.

1 reference

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7 January 2021

Stereoselective sulfation of terbutaline by the rat liver cytosol: evaluation of experimental approaches

1 reference

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7 January 2021

Pharmacokinetic evaluation in man of terbutaline given as separate enantiomers and as the racemate

1 reference

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7 January 2021

Pharmacokinetics of the enantiomers of terbutaline after repeated oral dosing with racemic terbutaline

1 reference

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7 January 2021

Racemates versus enantiomers in drug development: dogmatism or pragmatism?

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Salbutamol enantiomers: early clinical evidence in humans

1 reference

https://api.crossref.org/works/10.1016%2FS0091-6749%2899%2970414-8

7 January 2021

Effect of inhaled formoterol and budesonide on exacerbations of asthma. Formoterol and Corticosteroids Establishing Therapy (FACET) International Study Group.

1 reference

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7 January 2021

Comparison of addition of salmeterol to inhaled steroids with doubling of the dose of inhaled steroids

1 reference

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7 January 2021

10.1016/S0091-6749(99)70414-8

Identifiers

DOI

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release_4v7dmdeqkrhrrbw3tl4dje7a34

28 July 2017

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Fatcat

https://api.fatcat.wiki/v0/release/4v7dmdeqkrhrrbw3tl4dje7a34

24 November 2022

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PubMed ID

10329804

1 reference

PubMed ID

10329804