Synthesis and characterization of in vitro and in vivo profiles of hydroxybupropion analogues: aids to smoking cessation. (Q33955964)

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3 February 2020

title

Synthesis and characterization of in vitro and in vivo profiles of hydroxybupropion analogues: aids to smoking cessation (English)

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3 February 2020

7

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3 February 2020

author name string

Ronald J Lukas

1

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3 February 2020

Ana Z Muresan

2

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3 February 2020

M Imad Damaj

3

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3 February 2020

Bruce E Blough

4

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3 February 2020

Xiaodong Huang

5

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3 February 2020

Hernán A Navarro

6

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3 February 2020

J Brek Eaton

8

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3 February 2020

Syndia K Marxer-Miller

9

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3 February 2020

F Ivy Carroll

10

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3 February 2020

language of work or name

English

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publication date

1 June 2010

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Journal of Medicinal Chemistry

3 February 2020

published in

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3 February 2020

volume

53

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issue

12

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3 February 2020

page(s)

4731-4748

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Synthesis and biological evaluation of bupropion analogues as potential pharmacotherapies for smoking cessation.

3 February 2020

cites work

1 reference

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Effect of increasing intraperitoneal infusion rates on bupropion hydrochloride-induced seizures in mice

5 July 2018

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5 July 2018

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5 July 2018

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Bupropion for major depressive disorder: Pharmacokinetic and formulation considerations

5 July 2018

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Enantioselective effects of hydroxy metabolites of bupropion on behavior and on function of monoamine transporters and nicotinic receptors

5 July 2018

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Characterization of human alpha 4 beta 2-nicotinic acetylcholine receptors stably and heterologously expressed in native nicotinic receptor-null SH-EP1 human epithelial cells

5 July 2018

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Behavioral and biochemical investigations of bupropion metabolites

5 July 2018

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The diversity of subunit composition in nAChRs: evolutionary origins, physiologic and pharmacologic consequences

5 July 2018

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Pharmacokinetic optimisation of sustained-release bupropion for smoking cessation

5 July 2018

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Local anesthetics noncompetitively inhibit function of four distinct nicotinic acetylcholine receptor subtypes

5 July 2018

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Validation of bupropion hydroxylation as a selective marker of human cytochrome P450 2B6 catalytic activity.

5 July 2018

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CYP2B6 mediates the in vitro hydroxylation of bupropion: potential drug interactions with other antidepressants.

5 July 2018

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Reduced antinociception in mice lacking neuronal nicotinic receptor subunits

5 July 2018

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Characteristics of drug interactions with recombinant biogenic amine transporters expressed in the same cell type

5 July 2018

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Neuronal nicotinic receptor alpha 6 subunit mRNA is selectively concentrated in catecholaminergic nuclei of the rat brain

5 July 2018

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Characterization of nicotine binding in mouse brain and comparison with the binding of alpha-bungarotoxin and quinuclidinyl benzilate.

5 July 2018

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Synthesis and evaluation of furan, thiophene, and azole bis[(carbamoyloxy)methyl] derivatives as potential antineoplastic agents

5 July 2018

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The mesolimbic dopaminergic system is implicated in the reinforcing effects of nicotine

5 July 2018

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Calcium permeability and modulation of nicotinic acetylcholine receptor-channels in rat parasympathetic neurons

5 July 2018

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Stereoselective bupropion hydroxylation as an in vivo phenotypic probe for cytochrome P4502B6 (CYP2B6) activity

5 July 2018

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Smoking-induced ventral striatum dopamine release

29 October 2018

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Evaluation of the contribution of cytochrome P450 3A4 to human liver microsomal bupropion hydroxylation

29 October 2018

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29 October 2018

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29 October 2018

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(2S,3S,5R)-2-(3,5-difluorophenyl)-3,5-dimethyl-2-morpholinol: a novel antidepressant agent and selective inhibitor of norepinephrine uptake

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20509659

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM1003232

1 reference

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3 February 2020

1 reference

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3 February 2020

PubMed publication ID

20509659

1 reference