Identification of ML204, a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels (Q33973423)

30 July 2017

title

Identification of ML204, a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels (English)

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30 July 2017

15

Craig W Lindsley

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30 July 2017

Melissa Miller

1

1 reference

30 July 2017

Jie Shi

2

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30 July 2017

Yingmin Zhu

3

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30 July 2017

Maksym Kustov

4

1 reference

30 July 2017

Jin-bin Tian

5

1 reference

30 July 2017

Amy Stevens

6

1 reference

30 July 2017

Meng Wu

7

1 reference

30 July 2017

Jia Xu

8

1 reference

30 July 2017

Shunyou Long

9

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30 July 2017

Pu Yang

10

1 reference

30 July 2017

Alexander V Zholos

11

1 reference

30 July 2017

James M Salovich

12

1 reference

30 July 2017

C David Weaver

13

1 reference

30 July 2017

Corey R Hopkins

14

1 reference

30 July 2017

Owen McManus

16

1 reference

30 July 2017

Min Li

17

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30 July 2017

Michael X Zhu

18

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30 July 2017

language of work or name

English

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publication date

27 July 2011

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Journal of Biological Chemistry

30 July 2017

published in

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30 July 2017

volume

286

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30 July 2017

issue

38

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30 July 2017

page(s)

33436-33446

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Activation of TRP channels by protons and phosphoinositide depletion in Drosophila photoreceptors.

30 July 2017

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Activation of TRPA1 channels by fenamate nonsteroidal anti-inflammatory drugs

5 July 2018

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TRPC5 is a Ca2+-activated channel functionally coupled to Ca2+-selective ion channels

5 July 2018

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Deletion of TRPC4 and TRPC6 in mice impairs smooth muscle contraction and intestinal motility in vivo.

5 July 2018

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Intracellular calcium strongly potentiates agonist-activated TRPC5 channels.

5 July 2018

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The specific activation of TRPC4 by Gi protein subtype

5 July 2018

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Isoform-specific inhibition of TRPC4 channel by phosphatidylinositol 4,5-bisphosphate

5 July 2018

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Corticolimbic expression of TRPC4 and TRPC5 channels in the rodent brain

5 July 2018

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TRPC3 and TRPC4 associate to form a redox-sensitive cation channel. Evidence for expression of native TRPC3-TRPC4 heteromeric channels in endothelial cells.

5 July 2018

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Functional role of TRPC proteins in native systems: implications from knockout and knock-down studies.

5 July 2018

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Molecular analysis of a store-operated and 2-acetyl-sn-glycerol-sensitive non-selective cation channel. Heteromeric assembly of TRPC1-TRPC3.

5 July 2018

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Non-selective cationic channels of smooth muscle and the mammalian homologues of Drosophila TRP.

5 July 2018

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Human TRPC5 channel activated by a multiplicity of signals in a single cell

5 July 2018

1 reference

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2-aminoethoxydiphenyl borate is a common activator of TRPV1, TRPV2, and TRPV3

5 July 2018

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G-protein-gated TRP-like cationic channel activated by muscarinic receptors: effect of potential on single-channel gating

5 July 2018

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Contribution of transient receptor potential channels to the control of GABA release from dendrites

5 July 2018

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TRP channels as cellular sensors

5 July 2018

1 reference

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Homer Binds TRPC Family Channels and Is Required for Gating of TRPC1 by IP3 Receptors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Formation of novel TRPC channels by complex subunit interactions in embryonic brain

5 July 2018

1 reference

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TRPC4 and TRPC5: receptor-operated Ca2+-permeable nonselective cation channels

5 July 2018

1 reference

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Lanthanides potentiate TRPC5 currents by an action at extracellular sites close to the pore mouth

5 July 2018

1 reference

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Subunit composition of mammalian transient receptor potential channels in living cells

5 July 2018

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The TRP channels, a remarkably functional family

5 July 2018

1 reference

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The transient receptor potential protein homologue TRP6 is the essential component of vascular alpha(1)-adrenoceptor-activated Ca(2+)-permeable cation channel

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Lack of an endothelial store-operated Ca2+ current impairs agonist-dependent vasorelaxation in TRP4-/- mice

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Coassembly of Trp1 and Trp3 proteins generates diacylglycerol- and Ca2+-sensitive cation channels

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Receptor-mediated regulation of the nonselective cation channels TRPC4 and TRPC5.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Direct activation of human TRPC6 and TRPC3 channels by diacylglycerol

5 July 2018

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A novel capacitative calcium entry channel expressed in excitable cells

5 July 2018

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Muscarinic receptor subtypes controlling the cationic current in guinea-pig ileal smooth muscle.

5 July 2018

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Cloning and expression of a novel mammalian homolog of Drosophila transient receptor potential (Trp) involved in calcium entry secondary to activation of receptors coupled by the Gq class of G protein

5 July 2018

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SK&F 96365, a novel inhibitor of receptor-mediated calcium entry

5 July 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Intracellular calcium ions modulate acetylcholine-induced inward current in guinea-pig ileum

5 July 2018

1 reference

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Ins(1,4,5)P3 interacts with PIP2 to regulate activation of TRPC6/C7 channels by diacylglycerol in native vascular myocytes.

5 July 2018

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Crossref

https://api.crossref.org/works/10.1074%2FJBC.M111.274167

TRPC4 is an essential component of the nonselective cation channel activated by muscarinic stimulation in mouse visceral smooth muscle cells

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3190871

Impairment of store-operated Ca2+ entry in TRPC4(-/-) mice interferes with increase in lung microvascular permeability

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21795696

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Potentiating actions of lanthanum on ACh-induced cation current in guinea-pig ileal smooth muscle cells

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21795696

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Production of dissociated sensory neuron cultures and considerations for their use in studying neuronal function and plasticity

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21795696

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M111.274167

1 reference

30 July 2017

1 reference

30 July 2017

1 reference