Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs (Q34033184)

30 July 2017

title

Highly efficient synthesis and characterization of the GPR30-selective agonist G-1 and related tetrahydroquinoline analogs (English)

1 reference

30 July 2017

Cristian Bologa

5

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Eric R Prossnitz

object named as

Eric R Prossnitz

8

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Tudor I Oprea

object named as

Tudor Oprea

7

0 references

Larry Sklar

6

object named as

Larry A Sklar

1 reference

30 July 2017

Ritwik Burai

1

1 reference

30 July 2017

Chinnasamy Ramesh

2

1 reference

30 July 2017

Marvin Shorty

3

1 reference

30 July 2017

Ramona Curpan

4

1 reference

30 July 2017

Jeffrey B Arterburn

9

1 reference

30 July 2017

publication date

16 March 2010

1 reference

Organic and Biomolecular Chemistry

30 July 2017

published in

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30 July 2017

volume

8

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30 July 2017

issue

9

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30 July 2017

page(s)

2252-2259

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A crowdsourcing evaluation of the NIH chemical probes

30 July 2017

cites work

1 reference

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In vivo effects of a GPR30 antagonist

5 July 2018

1 reference

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Chronic treatment with the G protein-coupled receptor 30 agonist G-1 decreases blood pressure in ovariectomized mRen2.Lewis rats.

5 July 2018

1 reference

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Membrane estrogen receptor regulates experimental autoimmune encephalomyelitis through up-regulation of programmed death 1.

5 July 2018

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Rapid action of oestrogen in luteinising hormone-releasing hormone neurones: the role of GPR30.

5 July 2018

1 reference

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Regulatory role of G protein-coupled estrogen receptor for vascular function and obesity

5 July 2018

1 reference

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Involvement of G protein-coupled receptor 30 (GPR30) in rapid action of estrogen in primate LHRH neurons

5 July 2018

1 reference

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Expression of estrogen receptor GPR30 in the rat spinal cord and in autonomic and sensory ganglia

5 July 2018

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Extra-nuclear estrogen receptor GPR30 regulates serotonin function in rat hypothalamus.

5 July 2018

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Involvement of estradiol-17beta and its membrane receptor, G protein coupled receptor 30 (GPR30) in regulation of oocyte maturation in zebrafish, Danio rario

5 July 2018

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Nuclear and extranuclear pathway inputs in the regulation of global gene expression by estrogen receptors

5 July 2018

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The novel estrogen receptor, G protein-coupled receptor 30, mediates the proliferative effects induced by 17beta-estradiol on mouse spermatogonial GC-1 cell line.

5 July 2018

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G protein-coupled receptor 30 localizes to the endoplasmic reticulum and is not activated by estradiol

5 July 2018

1 reference

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The roles of membrane estrogen receptor subtypes in modulating dopamine transporters in PC-12 cells

5 July 2018

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Epidermal growth factor induces G protein-coupled receptor 30 expression in estrogen receptor-negative breast cancer cells

5 July 2018

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The G protein-coupled receptor GPR30 inhibits human urothelial cell proliferation.

5 July 2018

1 reference

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Estrogen signaling characteristics of Atlantic croaker G protein-coupled receptor 30 (GPR30) and evidence it is involved in maintenance of oocyte meiotic arrest

5 July 2018

1 reference

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Association of the membrane estrogen receptor, GPR30, with breast tumor metastasis and transactivation of the epidermal growth factor receptor

5 July 2018

1 reference

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Estrogen signaling through the transmembrane G protein-coupled receptor GPR30.

5 July 2018

1 reference

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Rapid estrogen signaling in the brain

5 July 2018

1 reference

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GPR30 contributes to estrogen-induced thymic atrophy

5 July 2018

1 reference

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G protein-coupled receptor 30 (GPR30) mediates gene expression changes and growth response to 17beta-estradiol and selective GPR30 ligand G-1 in ovarian cancer cells

5 July 2018

1 reference

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Povarov reactions involving 3-aminocoumarins: synthesis of 1,2,3,4-tetrahydropyrido[2,3-c]coumarins and pyrido[2,3-c]coumarins.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2913306

Nonclassical estrogen modulation of presynaptic GABA terminals modulates calcium dynamics in gonadotropin-releasing hormone neurons.

29 October 2018

1 reference

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Potential role of G-protein-coupled receptor 30 (GPR30) in estradiol-17beta-stimulated IGF-I mRNA expression in bovine satellite cell cultures

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2913306

GPR30 estrogen receptor agonists induce mechanical hyperalgesia in the rat.

29 October 2018

1 reference

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Distribution and characterization of estrogen receptor G protein-coupled receptor 30 in the rat central nervous system

29 October 2018

1 reference

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Virtual and biomolecular screening converge on a selective agonist for GPR30.

29 October 2018

1 reference

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Nonradical zinc-Barbier reaction for diastereoselective synthesis of vicinal amino alcohols

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2913306

Straightforward access to a structurally diverse set of oxacyclic scaffolds through a four-component reaction.

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2913306

InCl(3)-catalyzed domino reaction of aromatic amines with cyclic enol ethers in water: a highly efficient synthesis of new 1,2,3,4-tetrahydroquinoline derivatives

29 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2913306

First asymmetric synthesis of quinoline derivatives by inverse electron demand (IED) Diels-Alder reaction using chiral Ti(IV) complex

29 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20401403

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Total synthesis of the alkaloids martinelline and martinellic acid via a hetero Diels-Alder multicomponent coupling reaction

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20401403

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Intramolecular hetero Diels-Alder (Povarov) approach to the synthesis of the alkaloids luotonin A and camptothecin

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20401403

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1039/C001307B

1 reference

30 July 2017

1 reference

30 July 2017

1 reference