Non-peptide macrocyclic histone deacetylase inhibitors derived from tricyclic ketolide skeleton (Q34075642)

30 July 2017

title

Non-peptide macrocyclic histone deacetylase inhibitors derived from tricyclic ketolide skeleton (English)

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30 July 2017

7

Milan Mrksich

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author name string

Sandra C Mwakwari

1

1 reference

30 July 2017

William Guerrant

2

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30 July 2017

Vishal Patil

3

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30 July 2017

Shabana I Khan

4

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30 July 2017

Babu L Tekwani

5

1 reference

30 July 2017

Zachary A Gurard-Levin

6

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30 July 2017

Adegboyega K Oyelere

8

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30 July 2017

language of work or name

English

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publication date

1 August 2010

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Journal of Medicinal Chemistry

30 July 2017

published in

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30 July 2017

volume

53

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30 July 2017

issue

16

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30 July 2017

page(s)

6100-6111

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A structure-activity relationship study of the antimalarial and antileishmanial activities of nonpeptide macrocyclic histone deacetylase inhibitors

30 July 2017

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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Histone deacetylase inhibitors repress macrophage migration inhibitory factor (MIF) expression by targeting MIF gene transcription through a local chromatin deacetylation.

5 July 2018

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28 October 2018

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28 October 2018

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28 October 2018

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Structural snapshots of human HDAC8 provide insights into the class I histone deacetylases

28 October 2018

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Nonpeptide luteinizing hormone-releasing hormone antagonists derived from erythromycin A: design, synthesis, and biological activity of cladinose replacement analogues

28 October 2018

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Histone Deacetylase Inhibitors

28 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2924451

A simple colorimetric method to screen drug cytotoxicity against Leishmania using the dye Alamar Blue

28 October 2018

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Regulation of activity of the transcription factor GATA-1 by acetylation

28 October 2018

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Design and evaluation of 'Linkerless' hydroxamic acids as selective HDAC8 inhibitors

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20669972

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Synthesis and antibacterial activity of the tricyclic ketolides TE-802 and its analogs

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20669972

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JM100507Q

1 reference

30 July 2017

1 reference

30 July 2017

1 reference