JWH018, a common constituent of 'Spice' herbal blends, is a potent and efficacious cannabinoid CB receptor agonist (Q34098234)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

title

JWH018, a common constituent of 'Spice' herbal blends, is a potent and efficacious cannabinoid CB receptor agonist (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

0 references

0 references

0 references

1

1 reference

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17 January 2020

Ken Mackie

series ordinal

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

author name string

Alex Straiker

series ordinal

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

John Huffman

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

language of work or name

English

0 references

publication date

22 January 2010

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

British Journal of Pharmacology

17 January 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

volume

160

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

issue

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

page(s)

585-593

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

Endocannabinoid-mediated control of synaptic transmission

17 January 2020

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5 July 2018

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Cannabinoid-induced presynaptic inhibition of glutamatergic EPSCs in substantia gelatinosa neurons of the rat spinal cord

5 July 2018

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Retrograde inhibition of presynaptic calcium influx by endogenous cannabinoids at excitatory synapses onto Purkinje cells

5 July 2018

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5 July 2018

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Influence of the N-1 alkyl chain length of cannabimimetic indoles upon CB(1) and CB(2) receptor binding

5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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5 July 2018

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'Spice' and other herbal blends: harmless incense or cannabinoid designer drugs?

21 January 2018

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Cannabinoids suppress synaptic input to neurones of the rat dorsal motor nucleus of the vagus nerve

21 January 2018

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Segregation of two endocannabinoid-hydrolyzing enzymes into pre- and postsynaptic compartments in the rat hippocampus, cerebellum and amygdala.

21 January 2018

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21 January 2018

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21 January 2018

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Endogenous cannabinoids mediate retrograde signals from depolarized postsynaptic neurons to presynaptic terminals

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Localization of diacylglycerol lipase-alpha around postsynaptic spine suggests close proximity between production site of an endocannabinoid, 2-arachidonoyl-glycerol, and presynaptic cannabinoid CB1 receptor.

21 January 2018

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21 January 2018

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28 October 2018

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28 October 2018

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Internalization and Recycling of the CB1 Cannabinoid Receptor

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20100276

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

The third transmembrane helix of the cannabinoid receptor plays a role in the selectivity of aminoalkylindoles for CB2, peripheral cannabinoid receptor

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20100276

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

CB1 cannabinoid receptors are enriched in the perisynaptic annulus and on preterminal segments of hippocampal GABAergic axons

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20100276

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1111/J.1476-5381.2009.00582.X

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20100276%20AND%20SRC:MED&resulttype=core&format=json

17 January 2020

1 reference