Pharmacological profile of SB-357134: a potent, selective, brain penetrant, and orally active 5-HT(6) receptor antagonist (Q34117799)

31 July 2017

title

Pharmacological profile of SB-357134: a potent, selective, brain penetrant, and orally active 5-HT(6) receptor antagonist (English)

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31 July 2017

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Tania O Stean

1

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31 July 2017

Warren D Hirst

2

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31 July 2017

David R Thomas

3

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Gary W Price

4

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31 July 2017

Derek Rogers

5

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31 July 2017

Graham Riley

6

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31 July 2017

Steven M Bromidge

7

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31 July 2017

Halina T Serafinowska

8

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Douglas R Smith

9

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Sarah Bartlett

10

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Nigel Deeks

11

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31 July 2017

Mark Duxon

12

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31 July 2017

Neil Upton

13

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31 July 2017

language of work or name

English

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publication date

1 April 2002

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Pharmacology, Biochemistry and Behavior

31 July 2017

published in

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31 July 2017

volume

71

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issue

4

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31 July 2017

page(s)

645-654

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Investigation of stretching behaviour induced by the selective 5-HT6 receptor antagonist, Ro 04-6790, in rats.

31 July 2017

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Phenyl benzenesulfonamides are novel and selective 5-HT6 antagonists: identification of N-(2,5-dibromo-3-fluorophenyl)-4-methoxy-3-piperazin-1-ylbenzenesulfonamide (SB-357134).

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In vivo effects of the 5-HT(6) antagonist SB-271046 on striatal and frontal cortex extracellular concentrations of noradrenaline, dopamine, 5-HT, glutamate and aspartate

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2-Substituted tryptamines: agents with selectivity for 5-HT(6) serotonin receptors

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Characterization of [(125)I]-SB-258585 binding to human recombinant and native 5-HT(6) receptors in rat, pig and human brain tissue

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6-Bicyclopiperazinyl-1-arylsulfonylindoles and 6-bicyclopiperidinyl-1-arylsulfonylindoles derivatives as novel, potent, and selective 5-HT6 receptor antagonists

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Chemical protection against ionizing radiation. I. Sampling methods for screening compounds in radiation protection studies with mice

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Cloning, characterization, and chromosomal localization of a human 5-HT6 serotonin receptor

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Effects of the 5-HT(6) receptor antagonist Ro 04-6790 on learning consolidation

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5-HT6 receptor antagonists enhance retention of a water maze task in the rat.

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Characterization of SB-271046: a potent, selective and orally active 5-HT(6) receptor antagonist

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A novel rat serotonin (5-HT6) receptor: molecular cloning, localization and stimulation of cAMP accumulation

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Effects of altered 5-ht6 expression in the rat: functional studies using antisense oligonucleotides

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Characterization of Ro 04-6790 and Ro 63-0563: potent and selective antagonists at human and rat 5-HT6 receptors

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N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonists

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Profile of SB-204269, a mechanistically novel anticonvulsant drug, in rat models of focal and generalized epileptic seizures

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Localization of serotonin subtype 6 receptor messenger RNA in the rat brain by in situ hybridization histochemistry

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A role for 5-ht6 receptors in retention of spatial learning in the Morris water maze.

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Identifiers

DOI

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31 July 2017

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