Discovery of 3-[2-(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide (AP24534), a potent, orally active pan-inhibitor of breakpoint cluster region-abelson (BCR-ABL) kinase includ (Q34118184)
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English | Discovery of 3-[2-(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide (AP24534), a potent, orally active pan-inhibitor of breakpoint cluster region-abelson (BCR-ABL) kinase includ |
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Discovery of 3-[2-(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide (AP24534), a potent, orally active pan-inhibitor of breakpoint cluster region-abelson (BCR-ABL) kinase includ (English)
1 reference
Wei-Sheng Huang
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Chester A Metcalf
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Raji Sundaramoorthi
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Yihan Wang
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Dong Zou
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R Mathew Thomas
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Xiaotian Zhu
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Lisi Cai
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David Wen
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Shuangying Liu
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Jan Romero
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Jiwei Qi
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Ingrid Chen
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Geetha Banda
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Scott P Lentini
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Sasmita Das
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Qihong Xu
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Jeff Keats
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Frank Wang
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Scott Wardwell
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Yaoyu Ning
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Joseph T Snodgrass
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Marc I Broudy
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Karin Russian
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Tianjun Zhou
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Lois Commodore
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Narayana I Narasimhan
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Qurish K Mohemmad
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John Iuliucci
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Victor M Rivera
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David C Dalgarno
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Tomi K Sawyer
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Tim Clackson
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William C Shakespeare
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Identifiers
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