Optimization of N-benzyl-benzoxazol-2-ones as receptor antagonists of macrophage migration inhibitory factor (MIF) (Q34127116)

31 July 2017

title

Optimization of N-benzyl-benzoxazol-2-ones as receptor antagonists of macrophage migration inhibitory factor (MIF) (English)

1 reference

31 July 2017

1 reference

6

Richard Bucala

1 reference

31 July 2017

7

William L Jorgensen

1 reference

31 July 2017

3

Sunilkumar Gandavadi

1 reference

31 July 2017

2

Lin Leng

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

20 June 2024

5

Zoe Cournia

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

20 June 2024

author name string

Xin Du

series ordinal

4

1 reference

31 July 2017

Alissa A. Hare

series ordinal

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

20 June 2024

language of work or name

English

0 references

publication date

3 August 2010

1 reference

full work available at URL

31 July 2017

https://europepmc.org/articles/pmc2939296?pdf=render

file format

Portable Document Format

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

https://www.ncbi.nlm.nih.gov/pmc/articles/pmid/20728358/?tool=EBI

20 June 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

https://www.ncbi.nlm.nih.gov/pmc/articles/pmid/20728358/pdf/?tool=EBI

20 June 2024

file format

Portable Document Format

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

https://europepmc.org/articles/PMC2939296

20 June 2024

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

https://europepmc.org/articles/PMC2939296?pdf=render

20 June 2024

file format

Portable Document Format

online access status

open access

content deliverer

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

https://doi.org/10.1016/j.bmcl.2010.07.129

20 June 2024

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20728358

https://api.elsevier.com/content/article/PII:S0960894X1001098X?httpAccept=text/xml

20 June 2024

1 reference

Crossref

https://api.crossref.org/works/10.1016/J.BMCL.2010.07.129

https://api.elsevier.com/content/article/PII:S0960894X1001098X?httpAccept=text/plain

20 June 2024

1 reference

Crossref

https://api.crossref.org/works/10.1016/J.BMCL.2010.07.129

Bioorganic & Medicinal Chemistry Letters

20 June 2024

published in

1 reference

31 July 2017

volume

20

1 reference

31 July 2017

issue

19

1 reference

31 July 2017

page(s)

5811-5814

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Fragment screening of inhibitors for MIF tautomerase reveals a cryptic surface binding site

31 July 2017

cites work

1 reference

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Efficient drug lead discovery and optimization

5 July 2018

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Structural and Kinetic Analyses of Macrophage Migration Inhibitory Factor Active Site Interactions † ‡

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Discovery of human macrophage migration inhibitory factor (MIF)-CD74 antagonists via virtual screening

5 July 2018

1 reference

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A Novel, Macrophage Migration Inhibitory Factor Suicide Substrate Inhibits Motility and Growth of Lung Cancer Cells

5 July 2018

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ERK inhibitors as a potential new therapy for rheumatoid arthritis

5 July 2018

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Inhibition of macrophage migration inhibitory factor or its receptor (CD74) attenuates growth and invasion of DU-145 prostate cancer cells

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

CD44 is the signaling component of the macrophage migration inhibitory factor-CD74 receptor complex

5 July 2018

1 reference

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Extra precision glide: docking and scoring incorporating a model of hydrophobic enclosure for protein-ligand complexes

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

MIF: a new cytokine link between rheumatoid arthritis and atherosclerosis

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Macrophage migration inhibitory factor: a critical component of autoimmune inflammatory diseases.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Molecular modeling of organic and biomolecular systems using BOSS and MCPRO.

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Potential energy functions for atomic-level simulations of water and organic and biomolecular systems

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

MIF signal transduction initiated by binding to CD74

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Macrophage migration inhibitory factor and the discovery of tautomerase inhibitors

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Inhibition of macrophage migration inhibitory factor (MIF) tautomerase and biological activities by acetaminophen metabolites

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Pro-1 of macrophage migration inhibitory factor functions as a catalytic base in the phenylpyruvate tautomerase activity

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Characterization of the role of the amino-terminal proline in the enzymatic activity catalyzed by macrophage migration inhibitory factor

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Purification, bioactivity, and secondary structure analysis of mouse and human macrophage migration inhibitory factor (MIF).

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

A tautomerase-null macrophage migration-inhibitory factor (MIF) gene knock-in mouse model reveals that protein interactions and not enzymatic activity mediate MIF-dependent growth regulation

5 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2939296

Ionization state and molecular docking studies for the macrophage migration inhibitory factor: the role of lysine 32 in the catalytic mechanism

28 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20728358

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

A most interesting factor

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20728358

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identification and characterization of novel classes of macrophage migration inhibitory factor (MIF) inhibitors with distinct mechanisms of action

series ordinal

22

1 reference

Crossref

https://api.crossref.org/works/10.1016/J.BMCL.2010.07.129

20 June 2024

Identifiers

1 reference

31 July 2017

1 reference

31 July 2017

1 reference