Functional characterization of the semisynthetic bile acid derivative INT-767, a dual farnesoid X receptor and TGR5 agonist. (Q34310071)

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7 February 2020

title

Functional characterization of the semisynthetic bile acid derivative INT-767, a dual farnesoid X receptor and TGR5 agonist (English)

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7 February 2020

11

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author name string

Giovanni Rizzo

1

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7 February 2020

Daniela Passeri

2

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Francesca De Franco

3

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Gianmario Ciaccioli

4

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7 February 2020

Loredana Donadio

5

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Giorgia Rizzo

6

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Stefano Orlandi

7

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7 February 2020

Bahman Sadeghpour

8

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Xiaoxin X Wang

9

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7 February 2020

Tao Jiang

10

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Mark Pruzanski

12

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Luciano Adorini

13

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publication date

14 July 2010

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7 February 2020

published in

Molecular Pharmacology

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7 February 2020

volume

78

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7 February 2020

page(s)

617-630

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7 February 2020

issue

4

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Discovery of 6alpha-ethyl-23(S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesity.

7 February 2020

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6 July 2018

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6 July 2018

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6 July 2018

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The farnesoid X receptor modulates adiposity and peripheral insulin sensitivity in mice

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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28 October 2018

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28 October 2018

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28 October 2018

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28 October 2018

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28 October 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/20631053

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

The adipocyte as an endocrine cell

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PubMed

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inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1124/MOL.110.064501

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release_ndbunslxkzhd7cy3nl6lf6iuce

7 February 2020

Fatcat ID

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Fatcat

https://api.fatcat.wiki/v0/release/ndbunslxkzhd7cy3nl6lf6iuce

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20631053%20AND%20SRC:MED&resulttype=core&format=json

7 February 2020

1 reference