Conversion of A3 adenosine receptor agonists into selective antagonists by modification of the 5'-ribofuran-uronamide moiety (Q34313641)

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9 January 2020

title

Conversion of A3 adenosine receptor agonists into selective antagonists by modification of the 5'-ribofuran-uronamide moiety (English)

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9 January 2020

8

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1

Zhan-Guo Gao

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7

Lak Shin Jeong

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5

Hyuk Woo Lee

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9 January 2020

2

Bhalchandra V Joshi

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9 January 2020

3

Athena M Klutz

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9 January 2020

author name string

Soo-Kyung Kim

series ordinal

4

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9 January 2020

Hea Ok Kim

series ordinal

6

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9 January 2020

language of work or name

English

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publication date

10 November 2005

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Bioorganic & Medicinal Chemistry Letters

9 January 2020

published in

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volume

16

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9 January 2020

issue

3

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9 January 2020

page(s)

596-601

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RADIOLABELING AND EFFICIENT SYNTHESIS OF TRITIATED 2-CHLORO-N(6)-(3-IODOBENZYL)ADENOSINE-5'-N-METHYLURON-AMIDE, A POTENT, SELECTIVE A3 ADENOSINE RECEPTOR AGONIST.

9 January 2020

cites work

1 reference

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Structure-activity relationships of 2-chloro-N6-substituted-4'-thioadenosine-5'-uronamides as highly potent and selective agonists at the human A3 adenosine receptor

6 July 2018

1 reference

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Progress in the pursuit of therapeutic adenosine receptor antagonists

6 July 2018

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The cross-species A3 adenosine-receptor antagonist MRS 1292 inhibits adenosine-triggered human nonpigmented ciliary epithelial cell fluid release and reduces mouse intraocular pressure

6 July 2018

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(N)-methanocarba 2,N6-disubstituted adenine nucleosides as highly potent and selective A3 adenosine receptor agonists.

6 July 2018

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Purine receptors: GPCR structure and agonist design

6 July 2018

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Structural determinants of efficacy at A3 adenosine receptors: modification of the ribose moiety.

6 July 2018

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Some quantitative uses of drug antagonists

6 July 2018

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N6-substituted D-4'-thioadenosine-5'-methyluronamides: potent and selective agonists at the human A3 adenosine receptor

6 July 2018

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N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors

6 July 2018

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Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist

6 July 2018

1 reference

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2,5'-Disubstituted adenosine derivatives: evaluation of selectivity and efficacy for the adenosine A(1), A(2A), and A(3) receptor

6 July 2018

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International Union of Pharmacology. XXV. Nomenclature and classification of adenosine receptors

6 July 2018

1 reference

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Comparison of the potency of adenosine as an agonist at human adenosine receptors expressed in Chinese hamster ovary cells

6 July 2018

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A novel class of adenosine A3 receptor ligands. 2. Structure affinity profile of a series of isoquinoline and quinazoline compounds

6 July 2018

1 reference

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Derivatives of the triazoloquinazoline adenosine antagonist (CGS15943) are selective for the human A3 receptor subtype

6 July 2018

1 reference

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Structure-activity relationships of adenosine A3 receptor ligands: new potential therapy for the treatment of glaucoma

6 July 2018

1 reference

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Modeling the adenosine receptors: comparison of the binding domains of A2A agonists and antagonists

28 October 2018

1 reference

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Structural determinants of A(3) adenosine receptor activation: nucleoside ligands at the agonist/antagonist boundary

28 October 2018

1 reference

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Synthesis, biological activity, and molecular modeling investigation of new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives as human A(3) adenosine receptor antagonists

28 October 2018

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10.1016/J.BMCL.2005.10.054

28 October 2018

Identifiers

DOI

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9 January 2020

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9 January 2020

PubMed publication ID

16289820

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