An oral TRPV1 antagonist attenuates laser radiant-heat-evoked potentials and pain ratings from UV(B)-inflamed and normal skin (Q34330887)

1 August 2017

title

An oral TRPV1 antagonist attenuates laser radiant-heat-evoked potentials and pain ratings from UV(B)-inflamed and normal skin (English)

1 reference

1 August 2017

Ahmed A Othman

5

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Peter W. Reeh

object named as

Peter Reeh

2

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author name string

Klaus Schaffler

1

1 reference

1 August 2017

W Rachel Duan

3

1 reference

1 August 2017

Andrea E Best

4

1 reference

1 August 2017

Connie R Faltynek

6

1 reference

1 August 2017

Charles Locke

7

1 reference

1 August 2017

Wolfram Nothaft

8

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1 August 2017

language of work or name

English

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publication date

1 February 2013

1 reference

British Journal of Clinical Pharmacology

1 August 2017

published in

1 reference

1 August 2017

volume

75

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1 August 2017

issue

2

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1 August 2017

page(s)

404-414

1 reference

Guide to Receptors and Channels (GRAC), 5th edition

1 August 2017

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6 July 2018

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6 July 2018

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TRPV1: on the road to pain relief

6 July 2018

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6 July 2018

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TRPV1 controls acid- and heat-induced calcitonin gene-related peptide release and sensitization by bradykinin in the isolated mouse trachea

6 July 2018

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6 July 2018

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Repeated dosing of ABT-102, a potent and selective TRPV1 antagonist, enhances TRPV1-mediated analgesic activity in rodents, but attenuates antagonist-induced hyperthermia

6 July 2018

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(R)-(5-tert-butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)-urea (ABT-102) blocks polymodal activation of transient receptor potential vanilloid 1 receptors in vitro and heat-evoked firing of spinal dorsal horn neurons in vivo

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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Identification of (R)-1-(5-tert-butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea (ABT-102) as a potent TRPV1 antagonist for pain management

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21 January 2018

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21 January 2018

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PubMed

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inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1111/J.1365-2125.2012.04377.X

1 reference

1 August 2017

1 reference

1 August 2017

1 reference