Nature of pharmacophore influences active site specificity of proteasome inhibitors (Q34401062)

1 August 2017

title

Nature of pharmacophore influences active site specificity of proteasome inhibitors (English)

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1 August 2017

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ChEBI release 2020-05-28

Paul P Geurink

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Martijn Verdoes

object named as

Martijn Verdoes

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Bogdan I Florea

object named as

Bogdan I Florea

9

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Herman S Overkleeft

object named as

Herman S Overkleeft

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author name string

Michael Screen

1

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1 August 2017

Matthew Britton

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1 August 2017

Sondra L Downey

3

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1 August 2017

Mathias J Voges

5

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1 August 2017

Annet E M Blom

6

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1 August 2017

Martijn D P Risseeuw

8

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1 August 2017

Wouter A van der Linden

10

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1 August 2017

Alexandre A Pletnev

11

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1 August 2017

Alexei F Kisselev

13

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1 August 2017

language of work or name

English

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publication date

11 October 2010

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Journal of Biological Chemistry

1 August 2017

published in

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1 August 2017

volume

285

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1 August 2017

issue

51

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1 August 2017

page(s)

40125-40134

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A panel of subunit-selective activity-based proteasome probes

1 August 2017

cites work

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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21 January 2018

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21 January 2018

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The sizes of peptides generated from protein by mammalian 26 and 20 S proteasomes. Implications for understanding the degradative mechanism and antigen presentation

21 January 2018

1 reference

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https://pubmed.ncbi.nlm.nih.gov/20937826

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Importance of the different proteolytic sites of the proteasome and the efficacy of inhibitors varies with the protein substrate

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20937826

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M110.160606

1 reference

1 August 2017

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1 August 2017

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