The estradiol pharmacophore: ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site (Q34419702)

2 August 2017

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title

The estradiol pharmacophore: ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site (English)

1 reference

2 August 2017

Anstead GM

1

1 reference

PubMed ID

9071738

2 August 2017

Carlson KE

series ordinal

2

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PubMed ID

9071738

2 August 2017

Katzenellenbogen JA

series ordinal

3

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2 August 2017

1 March 1997

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2 August 2017

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2 August 2017

62

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2 August 2017

3

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2 August 2017

268-303

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2 August 2017

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7 January 2021

Binding, X-ray and NMR studies of the three A-ring isomers of natural estradiol

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A synthesis of 7 alpha-substituted estradiols: synthesis and biological evaluation of a 7 alpha-pentyl-substituted BODIPY fluorescent conjugate and a fluorine-18-labeled 7 alpha-pentylestradiol analog

1 reference

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7 January 2021

Synthesis and structure-affinity of a series of 7 alpha-undecylestradiol derivatives: a potential vector for therapy and imaging of estrogen-receptor-positive cancers

1 reference

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7 January 2021

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1 reference

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7 January 2021

ICI 182,780, a new antioestrogen with clinical potential

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7 January 2021

Studies with steroid-fluorescein conjugates on oestrogen target tissues

1 reference

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7 January 2021

Steroid structure and function--IX. Molecular conformation and receptor binding of isomeric analogs of D-homo-estradiol

1 reference

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7 January 2021

Quantitative structure-activity relationships of estrogenic steroids substituted at C14, C15

1 reference

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7 January 2021

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1 reference

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7 January 2021

Principles of protein-protein recognition

1 reference

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7 January 2021

Displacement of Estradiol from Estrogen Receptors by Simple Alkyl Phenols*

1 reference

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7 January 2021

Computer-aided drug design

1 reference

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7 January 2021

Seco-oestradiols and some non-steroidal oestrogens: Structural correlates of oestrogenic action

1 reference

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7 January 2021

Synthesis and biological activity of some 15-oxaestranes

1 reference

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7 January 2021

Identification of thiol group at the estrogen-binding site on the cytoplasmic receptor from rabbit uterus by affinity labeling

1 reference

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7 January 2021

Sulfhydryl Groups and Estradiol-Receptor Interaction

1 reference

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7 January 2021

Cysteinyl-tRNA synthetase from Escherichia coli does not need an editing mechanism to reject serine and alanine. High binding energy of small groups in specific molecular interactions

1 reference

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7 January 2021

Identification of amino acids in the hormone binding domain of the human estrogen receptor important in estrogen binding

1 reference

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7 January 2021

Carboxymethylation of the human estrogen receptor ligand-binding domain-estradiol complex: HPLC/ESMS peptide mapping shows that cysteine 447 does not react with iodoacetic acid

1 reference

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7 January 2021

Binding Activity of Oestrogen Receptors destroyed by Iodination

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7 January 2021

Differential inhibition of estrogen and antiestrogen binding to the estrogen receptor by diethylpyrocarbonate

1 reference

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7 January 2021

Differential interactions of estrogens and antiestrogens at the 17 beta-hydroxy or counterpart function with the estrogen receptor

1 reference

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7 January 2021

Evidence for involvement of tyrosine in estradiol binding by rat uterus estrogen receptor

1 reference

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7 January 2021

Contribution of hydrogen bonding to the conformational stability of ribonuclease T1

1 reference

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7 January 2021

Properties of a purified estradiol-dependent calf uterus tyrosine kinase

1 reference

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7 January 2021

Quantitative structure-activity relationships/comparative molecular field analysis (QSAR/CoMFA) for receptor-binding properties of halogenated estradiol derivatives

1 reference

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7 January 2021

Molecular structures, conformational analysis, and preferential modes of binding of 3-aroyl-2-arylbenzo[b]thiophene estrogen receptor ligands: LY117018 and aryl azide photoaffinity labeling analogs

1 reference

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7 January 2021

A MATHEMATICAL CONTRIBUTION TO STRUCTURE-ACTIVITY STUDIES.

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7 January 2021

Flexible Drug Molecules and Dynamic Receptors

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7 January 2021

Thermodynamic properties of ligand binding by monoclonal anti-fluorescyl antibodies.

1 reference

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7 January 2021

Molecular modelling of the human estrogen receptor and ligand interactions based on site-directed mutagenesis and amino acid sequence homology

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7 January 2021

A model for the determination of the 3D-spatial distribution of the functions of the hormone-binding domain of receptors that bind 3-keto-4-ene steroids

1 reference

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7 January 2021

Analysis of the binding of 3,3',5-triiodo-L-thyronine and its analogues to mutant human beta 1 thyroid hormone receptors: a model of the hormone binding site

1 reference

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7 January 2021

10.1016/S0039-128X(96)00242-5

Identifiers

DOI

1 reference

2 August 2017

1 reference

PubMed ID

9071738