Crystal Structures and Structure-Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors (Q34443476)

2 August 2017

title

Crystal Structures and Structure-Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors (English)

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2 August 2017

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Shingo Tojo

1

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2 August 2017

Tetsuya Kohno

2

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2 August 2017

Tomoyuki Tanaka

3

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2 August 2017

Seiji Kamioka

4

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2 August 2017

Yosuke Ota

5

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2 August 2017

Takayuki Ishii

6

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2 August 2017

Keiko Kamimoto

7

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2 August 2017

Shigehiro Asano

8

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2 August 2017

Yoshiaki Isobe

9

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2 August 2017

publication date

21 August 2014

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ACS Medicinal Chemistry Letters

2 August 2017

published in

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2 August 2017

volume

5

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2 August 2017

issue

10

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2 August 2017

page(s)

1119-1123

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Kynurenines in the CNS: recent advances and new questions.

2 August 2017

cites work

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6 July 2018

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6 July 2018

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Challenges and opportunities for new protein crystallization strategies in structure-based drug design

6 July 2018

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6 July 2018

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Structure based development of phenylimidazole-derived inhibitors of indoleamine 2,3-dioxygenase

6 July 2018

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6 July 2018

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6 July 2018

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Molecular insights into substrate recognition and catalysis by tryptophan 2,3-dioxygenase

6 July 2018

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Crystal structure of human indoleamine 2,3-dioxygenase: catalytic mechanism of O2 incorporation by a heme-containing dioxygenase

6 July 2018

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Biochemical and medical aspects of the indoleamine 2,3-dioxygenase-initiated L-tryptophan metabolism

6 July 2018

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Tryptophan degradation in mice initiated by indoleamine 2,3-dioxygenase

6 July 2018

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1-Methyl-DL-tryptophan, beta-(3-benzofuranyl)-DL-alanine (the oxygen analog of tryptophan), and beta-[3-benzo(b)thienyl]-DL-alanine (the sulfur analog of tryptophan) are competitive inhibitors for indoleamine 2,3-dioxygenase

6 July 2018

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Discovery of potent competitive inhibitors of indoleamine 2,3-dioxygenase with in vivo pharmacodynamic activity and efficacy in a mouse melanoma model.

6 July 2018

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High-level production of heme-containing holoproteins in Escherichia coli

27 October 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/25313323

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML500247W

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2 August 2017

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2 August 2017

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