N-Benzyl-5-methoxytryptamines as Potent Serotonin 5-HT2 Receptor Family Agonists and Comparison with a Series of Phenethylamine Analogues (Q34455931)

2 August 2017

N-Benzyl-5-methoxytryptamines as Potent Serotonin 5-HT2 Receptor Family Agonists and Comparison with a Series of Phenethylamine Analogues (English)

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2 August 2017

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5

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12 June 2020

author name string

David E Nichols

1

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12 June 2020

M Flori Sassano

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12 June 2020

Adam L Halberstadt

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12 June 2020

Landon M Klein

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12 June 2020

Simon P Elliott

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12 June 2020

Wolfgang J Fiedler

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publication date

21 January 2015

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ACS Chemical Neuroscience

2 August 2017

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12 June 2020

volume

6

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issue

7

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page(s)

1165-1175

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Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT₂A receptors, in mice

12 June 2020

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Interaction of 5-HT2A and 5-HT2C receptors in R(-)-2,5-dimethoxy-4-iodoamphetamine-elicited head twitch behavior in mice

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The serotonin 2C receptor potently modulates the head-twitch response in mice induced by a phenethylamine hallucinogen

6 July 2018

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A selective positive allosteric modulator of metabotropic glutamate receptor subtype 2 blocks a hallucinogenic drug model of psychosis

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Molecular interaction of serotonin 5-HT2A receptor residues Phe339(6.51) and Phe340(6.52) with superpotent N-benzyl phenethylamine agonists

6 July 2018

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Hallucinogen-like actions of 2,5-dimethoxy-4-(n)-propylthiophenethylamine (2C-T-7) in mice and rats

6 July 2018

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Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures(1).

6 July 2018

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N(1)-substituted ergolines and tryptamines show species differences for the agonist-labeled 5-HT2 receptor.

6 July 2018

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Species variations in transmembrane region V of the 5-hydroxytryptamine type 2A receptor alter the structure-activity relationship of certain ergolines and tryptamines

6 July 2018

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6 July 2018

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12 December 2020

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Identifiers

DOI

10.1021/CN500292D

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12 June 2020

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12 June 2020

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