CB2-selective cannabinoid receptor ligands: synthesis, pharmacological evaluation, and molecular modeling investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides (Q34525138)

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English	CB2-selective cannabinoid receptor ligands: synthesis, pharmacological evaluation, and molecular modeling investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides	scientific article

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scholarly article

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Europe PubMed Central

PubMed publication ID

2 August 2017

CB2-selective cannabinoid receptor ligands: synthesis, pharmacological evaluation, and molecular modeling investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides (English)

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Europe PubMed Central

PubMed publication ID

2 August 2017

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cannabinoid receptor

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Giuseppe Saccomanni

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Giuseppe Saccomanni

10

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Simone Bertini

4

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Mary E Abood

14

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Clementina Manera

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Clementina Manera

16

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Filippo Minutolo

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Filippo Minutolo

9

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Vincenzo Di Marzo

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Vincenzo Di Marzo

13

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Valentina Lucchesi

1

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2 August 2017

Dow P Hurst

2

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2 August 2017

Derek M Shore

3

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2 August 2017

Brandie M Ehrmann

5

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2 August 2017

Marco Allarà

6

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2 August 2017

Lyle Lawrence

7

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2 August 2017

Alessia Ligresti

8

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2 August 2017

Haleli Sharir

11

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2 August 2017

Marco Macchia

12

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2 August 2017

Patricia H Reggio

15

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2 August 2017

language of work or name

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publication date

15 October 2014

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2 August 2017

Journal of Medicinal Chemistry

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2 August 2017

57

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2 August 2017

21

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2 August 2017

8777-8791

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2 August 2017

describes a project that uses

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11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC4234427/fullTextXML

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Targeting the endocannabinoid system with cannabinoid receptor agonists: pharmacological strategies and therapeutic possibilities

1 reference

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Rational design, synthesis and anti-proliferative properties of new CB2 selective cannabinoid receptor ligands: an investigation of the 1,8-naphthyridin-2(1H)-one scaffold.

1 reference

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Crystal structure of metarhodopsin II

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A lipid pathway for ligand binding is necessary for a cannabinoid G protein-coupled receptor

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Conformational complexity of G-protein-coupled receptors

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Cysteine 2.59(89) in the second transmembrane domain of human CB2 receptor is accessible within the ligand binding crevice: evidence for possible CB2 deviation from a rhodopsin template.

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Identifiers

10.1021/JM500807E

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Europe PubMed Central

PubMed publication ID

2 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

2 August 2017

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