Inhibitors of type 5 17β-hydroxysteroid dehydrogenase (AKR1C3): overview and structural insights. (Q34618859)

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16 January 2020

title

Inhibitors of type 5 17β-hydroxysteroid dehydrogenase (AKR1C3): overview and structural insights (English)

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3

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author name string

Michael C Byrns

series ordinal

1

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16 January 2020

Yi Jin

series ordinal

2

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publication date

16 November 2010

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The Journal of Steroid Biochemistry and Molecular Biology

16 January 2020

published in

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16 January 2020

volume

125

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issue

1-2

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page(s)

95-104

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Human hydroxysteroid dehydrogenases and pre-receptor regulation: insights into inhibitor design and evaluation.

16 January 2020

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Intraprostatic androgens and androgen-regulated gene expression persist after testosterone suppression: therapeutic implications for castration-resistant prostate cancer

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An indomethacin analogue, N-(4-chlorobenzoyl)-melatonin, is a selective inhibitor of aldo-keto reductase 1C3 (type 2 3alpha-HSD, type 5 17beta-HSD, and prostaglandin F synthase), a potential target for the treatment of hormone dependent and hormone

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