The β-blocker Nebivolol Is a GRK/β-arrestin biased agonist (Q34972784)

5 August 2017

title

The β-blocker Nebivolol Is a GRK/β-arrestin biased agonist (English)

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5 August 2017

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7

Murat Bastepe

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5 August 2017

Catherine E Erickson

1

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5 August 2017

Rukhsana Gul

2

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5 August 2017

Christopher P Blessing

3

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5 August 2017

Jenny Nguyen

4

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5 August 2017

Tammy Liu

5

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5 August 2017

Lakshmi Pulakat

6

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5 August 2017

Edwin K Jackson

8

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5 August 2017

Bradley T Andresen

9

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5 August 2017

language of work or name

English

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publication date

20 August 2013

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5 August 2017

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5 August 2017

volume

8

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5 August 2017

issue

8

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5 August 2017

page(s)

e71980

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Creative Commons Attribution 4.0 International

5 August 2017

copyright license

start time

20 August 2013

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April 2022 Public Data File from Crossref

copyright status

copyrighted

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describes a project that uses

ImageJ

1 reference

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC3748024/fullTextXML

inferred from PubMed Central ID database lookup

cites work

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8 July 2018

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8 July 2018

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EGF receptor transactivation by G-protein-coupled receptors requires metalloproteinase cleavage of proHB-EGF

8 July 2018

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8 July 2018

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HL-1 cells: a cardiac muscle cell line that contracts and retains phenotypic characteristics of the adult cardiomyocyte

8 July 2018

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8 July 2018

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8 July 2018

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The receptor binding profile of the new antihypertensive agent nebivolol and its stereoisomers compared with various beta-adrenergic blockers

8 July 2018

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8 July 2018

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8 July 2018

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Human beta 1- and beta 2-adrenergic receptor binding and mediated accumulation of cAMP in transfected Chinese hamster ovary cells. Profile of nebivolol and known beta-adrenergic blockers

8 July 2018

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8 July 2018

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21 January 2018

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21 January 2018

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Nebivolol induces calcium-independent signaling in endothelial cells by a possible beta-adrenergic pathway

21 January 2018

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HB-EGF stimulates eNOS expression and nitric oxide production and promotes eNOS dependent angiogenesis.

21 January 2018

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21 January 2018

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Comparison of three radioligands for the labelling of human beta-adrenoceptor subtypes.

21 January 2018

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Nebivolol induces distinct changes in profibrosis microRNA expression compared with atenolol, in salt-sensitive hypertensive rats

21 January 2018

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Rational design and evaluation of new lead compound structures for selective betaARK1 inhibitors

21 January 2018

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Lack of evidence that nebivolol is a β₃-adrenoceptor agonist

21 January 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3748024

Assessment of nerve stimulation-induced release of purines from mouse kidneys by tandem mass spectrometry

26 October 2018

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Pharmacological and hemodynamic profile of nebivolol, a chemically novel, potent, and selective beta 1-adrenergic antagonist.

26 October 2018

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Energetics of Catalysis by Ribonucleases: Fate of the 2',3'-Cyclic Phosphodiester Intermediate

26 October 2018

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Epidermal growth factor (EGF) receptor-dependent ERK activation by G protein-coupled receptors: a co-culture system for identifying intermediates upstream and downstream of heparin-binding EGF shedding

21 January 2018

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12 December 2020

Studies on the mechanisms underlying beta-adrenoceptor-mediated relaxation of rat abdominal aorta

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12 December 2020

Beta-adrenoceptor-mediated cAMP accumulation in cardiac cells: effects of nebivolol

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12 December 2020

Nebivolol vasodilates human forearm vasculature: evidence for an L-arginine/NO-dependent mechanism

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12 December 2020

Carvedilol action is dependent on endogenous production of nitric oxide

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12 December 2020

10.1371/JOURNAL.PONE.0071980

Identifiers

DOI

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5 August 2017

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5 August 2017

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