Kinetics of Plasmodium falciparum thymidylate synthase: interactions with high-affinity metabolites of 5-fluoroorotate and D1694 (Q35125528)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8807052%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

title

Kinetics of Plasmodium falciparum thymidylate synthase: interactions with high-affinity metabolites of 5-fluoroorotate and D1694 (English)

1 reference

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19 October 2019

main subject

Plasmodium falciparum

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2

P K Rathod

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19 October 2019

author name string

M Hekmat-Nejad

series ordinal

1

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19 October 2019

language of work or name

English

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publication date

1 July 1996

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Antimicrobial Agents and Chemotherapy

19 October 2019

published in

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19 October 2019

volume

40

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19 October 2019

issue

7

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19 October 2019

page(s)

1628-1632

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Clonal viability measurements on Plasmodium falciparum to assess in vitro schizonticidal activity of leupeptin, chloroquine, and 5-fluoroorotate

19 October 2019

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13 July 2018

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13 July 2018

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Molecular cloning and sequence analysis of the Plasmodium falciparum dihydrofolate reductase-thymidylate synthase gene

13 July 2018

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Point mutations in the dihydrofolate reductase-thymidylate synthase gene as the molecular basis for pyrimethamine resistance in Plasmodium falciparum.

13 July 2018

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Selective activity of 5-fluoroorotic acid against Plasmodium falciparum in vitro

13 July 2018

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Expression of human thymidylate synthase in Escherichia coli

13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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ICI D1694, a quinazoline antifolate thymidylate synthase inhibitor that is a potent inhibitor of L1210 tumor cell growth in vitro and in vivo: a new agent for clinical study

13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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12 December 2020

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12 December 2020

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12 December 2020

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12 December 2020

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12 December 2020

Kinetic characteristics of ICI D1694: a quinazoline antifolate which inhibits thymidylate synthase

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12 December 2020

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Identifiers

DOI

10.1128/AAC.40.7.1628

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8807052%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:8807052%20AND%20SRC:MED&resulttype=core&format=json

19 October 2019

1 reference