Isothermal chemical denaturation to determine binding affinity of small molecules to G-protein coupled receptors (Q35163593)

6 August 2017

title

Isothermal chemical denaturation to determine binding affinity of small molecules to G-protein coupled receptors (English)

1 reference

G protein-coupled receptor

6 August 2017

main subject

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1 reference

Patrick Ross

1

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6 August 2017

Wilhelm Weihofen

2

1 reference

6 August 2017

Fai Siu

3

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6 August 2017

Amy Xie

4

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6 August 2017

Hetal Katakia

5

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6 August 2017

S Kirk Wright

6

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6 August 2017

Ian Hunt

7

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6 August 2017

Richard K Brown

8

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6 August 2017

Ernesto Freire

9

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6 August 2017

language of work or name

English

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publication date

4 December 2014

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6 August 2017

published in

Analytical Biochemistry

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6 August 2017

volume

473

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6 August 2017

page(s)

41-45

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Ligand binding analysis and screening by chemical denaturation shift

6 August 2017

cites work

1 reference

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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13 July 2018

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Thermodynamic stability of carbonic anhydrase: measurements of binding affinity and stoichiometry using ThermoFluor.

13 July 2018

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13 July 2018

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Unfolding free energy changes determined by the linear extrapolation method. 1. Unfolding of phenylmethanesulfonyl alpha-chymotrypsin using different denaturants

13 July 2018

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13 July 2018

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Analyzing ligand and small molecule binding activity of solubilized GPCRs using biosensor technology

27 September 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/25481736

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12 December 2020

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A high-throughput fluorescence chemical denaturation assay as a general screen for protein-ligand binding

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PubMed

https://pubmed.ncbi.nlm.nih.gov/25481736

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12 December 2020

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1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/25481736

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.AB.2014.11.019

1 reference

6 August 2017

1 reference

6 August 2017

1 reference